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Found 96 with Last Name = 'besra' and Initial = 'gs'
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50603476(CHEMBL5185220)
Affinity DataIC50:  221nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis DprE1 measured by resazurin dye based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574428(CHEMBL3262462)
Affinity DataIC50:  266nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574424(CHEMBL4858566)
Affinity DataIC50:  446nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574425(CHEMBL4877637)
Affinity DataIC50:  688nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574423(CHEMBL4873922)
Affinity DataIC50:  698nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574429(CHEMBL4857182)
Affinity DataIC50:  794nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574427(CHEMBL4848357)
Affinity DataIC50:  922nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148588(CHEMBL325304 | Heptyl-phosphonic acid monoethyl es...)
Affinity DataIC50:  1.06E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148588(CHEMBL325304 | Heptyl-phosphonic acid monoethyl es...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148590((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148590((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  1.31E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148587(CHEMBL326268 | Heptyl-phosphonic acid mono-[2-(1,3...)
Affinity DataIC50:  1.47E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50603478(CHEMBL5197259)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50195746(CHEMBL227546 | ethyl 3-phenoxybenzyl butylphosphon...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148586(Butyl-phosphonic acid ethyl ester 3-phenoxy-benzyl...)
Affinity DataIC50:  2.01E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574426(CHEMBL4865471)
Affinity DataIC50:  2.16E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50220630(5-(4-methoxycarbonyl-biphenyl-4-ylmethyl)-4-hydrox...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50603476(CHEMBL5185220)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148593(CHEMBL119521 | Hexyl-phosphonic acid monoethyl est...)
Affinity DataIC50:  3.56E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148593(CHEMBL119521 | Hexyl-phosphonic acid monoethyl est...)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50220624(4'-(3-hydroxy-2,4-dimethyl-5-oxo-2,5-dihydro-thiop...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148585(CHEMBL418868 | Hexyl-phosphonic acid mono-[2-(1,3-...)
Affinity DataIC50:  4.39E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50220629(4'-(3-hydroxy-2,4-dimethyl-5-oxo-2,5-dihydro-thiop...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50603477(CHEMBL5205737)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148594((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148594((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50195743(CHEMBL427453 | ethyl 3-phenoxybenzyl nonylphosphon...)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148583(CHEMBL325149 | Nonyl-phosphonic acid ethyl ester 3...)
Affinity DataIC50:  1.48E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50220625(4-hydroxy-3,5-dimethyl-5-(4-phenoxy-benzyl)-5H-thi...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134362(5-(4'-Benzyloxymethyl-biphenyl-4-ylmethyl)-4-hydro...)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134348(4-Hydroxy-5-(4'-hydroxymethyl-biphenyl-4-ylmethyl)...)
Affinity DataIC50:  1.90E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50195748(CHEMBL227405 | ethyl 3-phenoxybenzyl heptylphospho...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148596(CHEMBL278017 | Heptyl-phosphonic acid ethyl ester ...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134356(5-(4'-tert-Butyl-biphenyl-4-ylmethyl)-4-hydroxy-3,...)
Affinity DataIC50:  2.50E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148582(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-ethylet...)
Affinity DataIC50:  2.57E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148582(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-ethylet...)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134352(4'-(3-Hydroxy-2,4-dimethyl-5-oxo-2,5-dihydro-thiop...)
Affinity DataIC50:  2.90E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50520740(CHEMBL4586075)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by whole-cell patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50603479(CHEMBL5187959)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148597((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyleth...)
Affinity DataIC50:  4.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148597((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyleth...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148584(CHEMBL118790 | Hexyl-phosphonic acid ethyl ester 3...)
Affinity DataIC50:  4.26E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50195749(CHEMBL223946 | ethyl 3-phenoxybenzyl hexylphosphon...)
Affinity DataIC50:  4.26E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham

Curated by ChEMBL
LigandPNGBDBM50134355(5-(4-tert-Butyl-benzyl)-4-hydroxy-3,5-dimethyl-5H-...)
Affinity DataIC50:  4.30E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50574428(CHEMBL3262462)
Affinity DataIC50:  4.79E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50520740(CHEMBL4586075)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50520740(CHEMBL4586075)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50520740(CHEMBL4586075)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50520740(CHEMBL4586075)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP1A2 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50520740(CHEMBL4586075)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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