TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 221nMAssay Description:Inhibition of recombinant Mycobacterium tuberculosis DprE1 measured by resazurin dye based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 266nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 446nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 688nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 698nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 794nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 922nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.06E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.31E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.47E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.01E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DprE1 using FAD as substrate by resazurin based assayMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 4.39E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by whole-cell patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 4.26E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobaterium tuberculosisMore data for this Ligand-Target Pair
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis)
University Of Ljubljana
Curated by ChEMBL
University Of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 4.26E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant antigen 85C mycolyltransferaseMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis)
University Of Birmingham
Curated by ChEMBL
University Of Birmingham
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:In vitro inhibitory activity against the recombinant Mycobacterium tuberculosis Beta-ketoacyl-ACP synthase III mtFabH condensing enzyme.More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 2C9(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 2C19(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 1A2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP1A2 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair