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Found 143 with Last Name = 'black' and Initial = 'rm'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157931(2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166292((S)-2-{3-[1-(4-Methoxy-phenyl)-2-methyl-5-trifluor...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157917((2S)-2-(3-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFL...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157933(2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157926(2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166300((S)-2-{2-Chloro-5-[1-(6-chloro-benzo[d]isoxazol-3-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166295((R)-2-{4-Chloro-3-[1-(6-methoxy-benzo[d]isoxazol-3...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157936((2S)-2-(2-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFL...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157917((2S)-2-(3-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFL...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157920(2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157927((R)-2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluo...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157925(2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157919(2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157921(2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166298((2S)-2-(4-chloro-3-(1-(6-chlorobenzo[d]isoxazol-3-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166302((S)-2-{5-[1-(6-Chloro-benzo[d]isoxazol-3-yl)-2-met...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157932((R)-2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluo...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166296((S)-2-{3-[1-(6-Methoxy-quinolin-3-yl)-2-methyl-5-t...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290785(CHEMBL406357 | Pneumocandin analogue)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166293((S)-2-{3-[1-(6-Chloro-benzo[d]isoxazol-3-yl)-2-met...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290778(CHEMBL414690 | Pneumocandin analogue)
Affinity DataIC50:  35nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290798(CHEMBL268721 | Pneumocandin analogue)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166303(CHEMBL191087 | {3-[1-(4-Methoxy-benzoyl)-2-methyl-...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157916(2-{3-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50:  45nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157934(2-{3-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50:  49nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166305((S)-2-[3-(2-Methyl-5-trifluoromethoxy-1H-indol-3-y...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration against Cytochrome P450 2C9 in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290784(CHEMBL413522 | Pneumocandin analogue)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290792(CHEMBL441213 | Pneumocandin analogue)
Affinity DataIC50:  60nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166301((4-Methoxy-phenyl)-[2-methyl-3-(3-prop-2-ynyloxy-b...)
Affinity DataIC50:  62nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290777(CHEMBL428264 | Pneumocandin analogue)
Affinity DataIC50:  70nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290797(CHEMBL267988 | Pneumocandin analogue)
Affinity DataIC50:  70nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290803(CHEMBL407395 | Pneumocandin analogue)
Affinity DataIC50:  70nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157918(2-{2-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50:  79nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290793(CHEMBL410837 | Pneumocandin analogue)
Affinity DataIC50:  80nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157930(2-{2-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50:  84nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157938(CHEMBL178562 | {4-[1-(4-Chloro-benzoyl)-5-methoxy-...)
Affinity DataIC50:  84nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290796(CHEMBL439260 | Pneumocandin analogue)
Affinity DataIC50:  90nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290801(CHEMBL384968 | Pneumocandin analogue)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290791(CHEMBL408285 | Pneumocandin analogue)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290775(CHEMBL415669 | Pneumocandin analogue)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166294((S)-2-{3-Chloro-5-[1-(6-chloro-benzo[d]isoxazol-3-...)
Affinity DataIC50:  109nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290782(CHEMBL385665 | Pneumocandin analogue)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166297((S)-2-{3-[1-(6-Methoxy-quinolin-2-yl)-2-methyl-5-t...)
Affinity DataIC50:  135nMAssay Description:Inhibition of human peroxisome proliferator activated receptor gamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290780(CHEMBL412195 | Pneumocandin analogue)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290788(CHEMBL438185 | Pneumocandin analogue)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290781(CHEMBL387275 | Pneumocandin analogue)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290789(CHEMBL408469 | Pneumocandin analogue)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
TBA

Curated by ChEMBL
LigandPNGBDBM50290783(CHEMBL386826 | Pneumocandin analogue)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of 1,3-beta-glucan synthase in Candida albicans membrane assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157929(3-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-indo...)
Affinity DataIC50:  208nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50481375(CHEMBL593032)
Affinity DataIC50:  230nMAssay Description:Inhibition of gamma secretase in human SHSY5Y cells expressing wild-type APP assessed as inhibition of intracellular amyloid beta-42 by electrochemil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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