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Found 39 with Last Name = 'blanchard' and Initial = 'je'
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50294336(5-amino-2-(4-aminophenylamino)benzenesulfonic acid...)
Affinity DataKi:  17nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50483325(CHEMBL1652297 | Mac0029665)
Affinity DataKi:  23nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50483326(CHEMBL1652296 | Mac0008028)
Affinity DataKi:  404nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370860(CHEMBL219268)
Affinity DataIC50:  79nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370870(CHEMBL218090)
Affinity DataIC50:  280nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370869(CHEMBL220764)
Affinity DataIC50:  530nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM68271(M-31850)
Affinity DataIC50:  600nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370861(CHEMBL221848)
Affinity DataIC50:  650nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370865(CHEMBL221706)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370853(CHEMBL221182)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370850(CHEMBL373750)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370867(CHEMBL221705)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370855(CHEMBL218737)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM68272(LU79953)
Affinity DataIC50:  4.60E+3nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84610(5-(3,5-dichlorophenoxy)-N-(4-pyrdinyl)-2- furamide...)
Affinity DataIC50:  4.70E+3nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370857(CHEMBL220531)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370854(CHEMBL220494)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370864(CHEMBL451558)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM18046(5-((4-methylphenyl)thio)-quinazoline 2,4-diamine, ...)
Affinity DataIC50:  7.80E+3nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370856(CHEMBL376005)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370866(CHEMBL219582)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370848(CHEMBL218058)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM68270(5141402)
Affinity DataIC50:  1.60E+4nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM50106194(1,3-dioxo-1H-benz[de]isoquinoline | 1,8-Naphthalim...)
Affinity DataIC50:  1.80E+4nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84609(7,8-diethoxy-quinazoline 2,4-diamine, 1b)
Affinity DataIC50:  2.20E+4nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370858(CHEMBL220530)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM68269(M-31867)
Affinity DataIC50:  3.10E+4nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370859(CHEMBL383877)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370852(CHEMBL219322)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370851(CHEMBL375564)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84608(2,4-diamino-6-nitro-quinazoline, 1a)
Affinity DataIC50:  6.10E+4nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84611(2-methyl-N-pyridin-4-yl-benzamide, 2a)
Affinity DataIC50:  8.00E+4nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370863(CHEMBL222116)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM68268(M-31862)
Affinity DataIC50:  1.08E+5nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit alpha(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM68267(M-31860)
Affinity DataIC50:  1.38E+5nMT: 2°CAssay Description:Enzyme assay based on 4-MU substrates with HTS to identify inhibitory compounds for Hex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370868(CHEMBL218485)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84612(2,2-dimethyl-N-(4-pyridinyl)propanamide, 2b)
Affinity DataIC50: >4.00E+5nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370849(CHEMBL385118)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystathionine beta-lyase MetC(Escherichia coli K-12)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50370862(CHEMBL221962)
Affinity DataIC50:  5.60E+5nMAssay Description:Inhibition of Escherichia coli CBLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed