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Found 182 with Last Name = 'bockaert' and Initial = 'j'
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000580nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000630nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.000870nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.000910nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.00560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.00890nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(5-Fluoro-2-methoxy-1H-indole-3-carboxylic acid [1-...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.470nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM86038(SL65.0155 | SL650155)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85019(4-Amino-5-chloro-N-(1-{4-[4-(dimethylamino)-1-pipe...)
Affinity DataKi:  1.38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85019(4-Amino-5-chloro-N-(1-{4-[4-(dimethylamino)-1-pipe...)
Affinity DataKi:  1.38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85019(4-Amino-5-chloro-N-(1-{4-[4-(dimethylamino)-1-pipe...)
Affinity DataKi:  2.88nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007863(6-Methoxy-2-oxo-2,3-dihydro-benzoimidazole-1-carbo...)
Affinity DataKi:  5.37nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056401(2-diethylaminoethyl [2-methoxy-4-amino-5-chloro]be...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056401(2-diethylaminoethyl [2-methoxy-4-amino-5-chloro]be...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056401(2-diethylaminoethyl [2-methoxy-4-amino-5-chloro]be...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056401(2-diethylaminoethyl [2-methoxy-4-amino-5-chloro]be...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50005833((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
Affinity DataKi:  7.41nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056401(2-diethylaminoethyl [2-methoxy-4-amino-5-chloro]be...)
Affinity DataKi:  7.76nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50005833((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50005833((exo)4-Amino-5-chloro-N-(hexahydro-pyrrolizin-1-yl...)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007863(6-Methoxy-2-oxo-2,3-dihydro-benzoimidazole-1-carbo...)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM84648(BIMU 8)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007863(6-Methoxy-2-oxo-2,3-dihydro-benzoimidazole-1-carbo...)
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056404(3-Isopropyl-2-oxo-2,3-dihydro-benzoimidazole-1-car...)
Affinity DataKi:  19.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate metabotropic receptor 5(PORCINE)
Cnrs Ccipe

Curated by PDSP Ki Database
LigandPNGBDBM17660((2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-2-yl...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007863(6-Methoxy-2-oxo-2,3-dihydro-benzoimidazole-1-carbo...)
Affinity DataKi:  22.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM84648(BIMU 8)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM84648(BIMU 8)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM84648(BIMU 8)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007863(6-Methoxy-2-oxo-2,3-dihydro-benzoimidazole-1-carbo...)
Affinity DataKi:  26.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(MOUSE)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007863(6-Methoxy-2-oxo-2,3-dihydro-benzoimidazole-1-carbo...)
Affinity DataKi:  26.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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