Affinity DataIC50: 1.32nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 8nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 16nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 20nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 30nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 44nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 45nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer upon incubation for 1 ...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 54nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 230nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair