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Found 12 with Last Name = 'boerman' and Initial = 'oc'
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318385(2-(4-{[(2-{[(3-{[1-(5-{[(1R)-1-{[(4R,7S,10S,13R,16...)
Affinity DataIC50:  1.32nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318386(2-[7-({[2-({[3,5-bis({[1-(5-{[(1R)-1-{[(4R,7S,10S,...)
Affinity DataIC50:  2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318388((4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-N-[(2R,3...)
Affinity DataIC50:  2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174609((LTB4-(Csa)4)2-Glu-H Conjugate | CHEMBL412510)
Affinity DataIC50:  8nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50318387(CHEMBL1099306)
Affinity DataIC50:  14nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174608(CHEMBL406432 | HYNIC Conjugate)
Affinity DataIC50:  16nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174610(2-[5-Methyl-5-(1H-tetrazol-5-yl)-hexyloxy]-4,6-dip...)
Affinity DataIC50:  20nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174607(CHEMBL415548 | DTPA Conjugate)
Affinity DataIC50:  30nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174606(CHEMBL384950 | HYNIC Analogue)
Affinity DataIC50:  44nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174606(CHEMBL384950 | HYNIC Analogue)
Affinity DataIC50:  45nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer upon incubation for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174607(CHEMBL415548 | DTPA Conjugate)
Affinity DataIC50:  54nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging

Curated by ChEMBL
LigandPNGBDBM50174611(CHEMBL437275 | HYNIC Conjugate)
Affinity DataIC50:  230nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed