Affinity DataKi: 220nM IC50: 30nMpH: 7.4Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in 10 mM phosphate-buffered saline (pH 7.4). IC50, defined as t...More data for this Ligand-Target Pair
Affinity DataKi: 560nM IC50: 320nMpH: 7.4Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in 10 mM phosphate-buffered saline (pH 7.4). IC50, defined as t...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nM IC50: 3.40E+3nMpH: 7.4Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in 10 mM phosphate-buffered saline (pH 7.4). IC50, defined as t...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nM IC50: 100nMpH: 7.4Assay Description:Steady state kinetics were performed on an Agilent 8453 diode array spectrophotometer in 10 mM phosphate-buffered saline (pH 7.4). IC50, defined as t...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:The concentration of compound to inhibit beta-lactamase was measured on E. coli WC3310More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of class A TEM-1 beta-lactamase derived from Enterobacter cloacaeMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Inhibitory activity against class A TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibitory activity against class A TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibitory activity against class A TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:The compound was evaluated for inhibition against Class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against class A TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:The compound was evaluated for inhibition against the GC1 extended spectrum Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of class A TEM-1 beta-lactamase derived from Enterobacter cloacaeMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against serine beta-lactamase, PC1 (class A) derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:The compound was evaluated for inhibition against the GC1 extended spectrum Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of class A TEM-1 beta-lactamase derived from Enterobacter cloacaeMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:The concentration of compound to inhibit beta-lactamase was measured on E. cloacae SC 12368More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:The concentration of compound to inhibit beta-lactamase was measured on Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:The concentration of compound to inhibit Beta-lactamase was measured on Escherichia coli WC3310More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae SC 12368 E-2More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Affinity for alpha4-beta1 integrin from HL60 cell lysateMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:The compound was evaluated for inhibition against Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of Class C beta-lactamase from E. cloacae strain P99More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibitory activity against class A TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:The concentration of compound to inhibit beta-lactamase was measured on E. coli WC3310More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair