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Found 43 with Last Name = 'campbell' and Initial = 'sj'
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380359(CHEMBL2017822)
Affinity DataKi:  40nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380358(CHEMBL2017821)
Affinity DataKi:  80nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380353(CHEMBL2017816)
Affinity DataKi:  100nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380352(CHEMBL2017815)
Affinity DataKi:  130nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50345641((S)-2-((S)-2-((S)-1-((S)-2-acetamido-3-(phosphonoo...)
Affinity DataKi:  200nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataKi:  270nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380354(CHEMBL2017817)
Affinity DataKi:  500nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380351(CHEMBL2017814)
Affinity DataKi:  540nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380349(CHEMBL2017812)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50345623((S)-2-acetamido-3-((S)-2-((2S,3R)-1-((S)-1-amino-1...)
Affinity DataKi:  1.85E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50345629((S)-2-acetamido-3-((S)-2-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataKi:  1.96E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380357(CHEMBL2017820)
Affinity DataKi:  4.04E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380355(CHEMBL2017818)
Affinity DataKi:  1.21E+4nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380356(CHEMBL2017819)
Affinity DataKi:  1.57E+4nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50380350(CHEMBL2017813)
Affinity DataKi:  1.94E+4nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050527(Boronic acid derivative | CHEMBL66032 | US11096924...)
Affinity DataIC50:  11nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  15nMAssay Description:Compound was tested in vitro for inhibition of Dipeptidylpeptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50:  15nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050521((2-Dihydroxyborane-pyrrolidin-1-yl)-pyrrolidin-2-y...)
Affinity DataIC50:  20nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  21nMAssay Description:Compound was tested in vitro for inhibition of Dipeptidylpeptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369128(CHEMBL1790483 | US11096924, DASH-inhibitors 4316 |...)
Affinity DataIC50:  25nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  26nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050514(Boronic acid derivative | CHEMBL304007)
Affinity DataIC50:  32nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
Affinity DataIC50:  44nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50:  60nMAssay Description:Compound was tested in vitro for inhibition of Dipeptidylpeptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050520(Boronic acid derivative | CHEMBL63406 | US11096924...)
Affinity DataIC50:  60nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050524(Boronic acid derivative | CHEMBL291428)
Affinity DataIC50:  63nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050515(Boronic acid derivative | CHEMBL63652 | US11096924...)
Affinity DataIC50:  70nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50:  95nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369129(CHEMBL1790478)
Affinity DataIC50:  190nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050526(Boronic acid derivative | CHEMBL292342)
Affinity DataIC50:  250nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369129(CHEMBL1790478)
Affinity DataIC50:  730nMAssay Description:Compound was tested in vitro for inhibition of Dipeptidylpeptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050521((2-Dihydroxyborane-pyrrolidin-1-yl)-pyrrolidin-2-y...)
Affinity DataIC50:  770nMAssay Description:Compound was tested in vitro for inhibition of Dipeptidylpeptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was tested in vitro for inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050512(Boronic acid derivative | CHEMBL65406)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369129(CHEMBL1790478)
Affinity DataIC50:  6.00E+3nMAssay Description:Compound was tested in vitro for inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050511((R)-1-(2-aminoacetyl)pyrrolidin-2-ylboronic acid |...)
Affinity DataIC50:  1.60E+4nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050519(Boronic acid derivative | CHEMBL303131)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050512(Boronic acid derivative | CHEMBL65406)
Affinity DataIC50:  1.80E+4nMAssay Description:Compound was tested in vitro for inhibition of Dipeptidylpeptidase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  2.30E+4nMAssay Description:Compound was tested in vitro for inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050523(Boronic acid derivative | CHEMBL66189)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  6.10E+4nMAssay Description:Compound was tested in vitro for inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  1.16E+5nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed