Affinity DataKi: 6.00E+4nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme activity at pH 8.5 in rabbit lungMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme activity at pH 8.5 in rabbit lungMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme activity at pH 8.5 in rabbit lungMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:In vitro inhibition of Angiotensin I converting enzyme activity at pH 8.5 in rabbit lungMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of DPP4 (unknown origin) pre-incubated for 1 hr before Gly-Pro-pNA substrate addition and measured 2 hrs post substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of DPP4 (unknown origin) pre-incubated for 1 hr before Gly-Pro-pNA substrate addition and measured 2 hrs post substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of DPP4 (unknown origin) pre-incubated for 1 hr before Gly-Pro-pNA substrate addition and measured 2 hrs post substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 269nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 295nMAssay Description:Inhibition of solubilized, purified rat liver HMG-CoA reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of Clostridium botulinum BoNT/A light chain using SNAPtide as substrate by FRET based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 348nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (morn)More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 363nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of DPP4 (unknown origin) pre-incubated for 1 hr before Gly-Pro-pNA substrate addition and measured 2 hrs post substrate additionMore data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 581nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 636nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Inhibition of DPP4 (unknown origin) pre-incubated for 1 hr before Gly-Pro-pNA substrate addition and measured 2 hrs post substrate additionMore data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 742nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (morn)More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Clostridium botulinum BoNT/A using SNAP-25 (66-mer) as substrate by LC-MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Collaborative Innovation Center Of Functionalized Probes For Chemical Imaging In University Of Shandong
Curated by ChEMBL
Collaborative Innovation Center Of Functionalized Probes For Chemical Imaging In University Of Shandong
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of bovine XOD assessed as inhibition of uric acid formation using xanthine as substrate preincubated with enzyme for 5 mins followed by su...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.54E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Collaborative Innovation Center Of Functionalized Probes For Chemical Imaging In University Of Shandong
Curated by ChEMBL
Collaborative Innovation Center Of Functionalized Probes For Chemical Imaging In University Of Shandong
Curated by ChEMBL
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of bovine XOD assessed as inhibition of uric acid formation using xanthine as substrate preincubated with enzyme for 5 mins followed by su...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of N-terminal 6XHis-tagged Clostridium botulinum BoNT/A light chain C-terminal truncation mutant (1 to 425 residues) expressed in Escheric...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals
Curated by ChEMBL
Enanta Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.92E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assay (MOM)More data for this Ligand-Target Pair