Affinity DataKi: 0.0200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:PKi was measured by Histamine H3 receptor binding assay (N-alpha-MeHA) on rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 79.4nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 199nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 199nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against prolyl oligopeptidase of porcine brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:In vitro inhibition of prolyl oligopeptidase (POP) from pig brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:In vitro inhibitory activity of the compound against prolyl oligopeptidase (POP) from pigbrain expressedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:In vitro inhibition of prolyl oligopeptidase (POP) from pig brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:In vitro inhibitory activity of the compound against prolyl oligopeptidase (POP) from pig brain ;value ranges from (1.1-2.2)More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:In vitro inhibition of prolyl oligopeptidase (POP) from pig brainMore data for this Ligand-Target Pair