TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of S-adenosyl-L-homocysteine hydrolase in intact rat hepatocytesMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of S-adenosyl-L-homocysteine hydrolase after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of S-adenosyl-L-homocysteine hydrolaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Affinity DataIC50: 3.21E+3nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.66E+3nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Affinity DataIC50: 2.45E+4nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of S-adenosyl-L-homocysteine hydrolase after 10 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of S-adenosyl-L-homocysteine hydrolase after 10 mins by scintillation countingMore data for this Ligand-Target Pair