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Found 78 with Last Name = 'cianetti' and Initial = 's'
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485494(CHEMBL2063089)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485491(CHEMBL2063088)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485492(Grazoprevir | Grazoprevir monohydrate | MK-5172 | ...)
Affinity DataKi:  0.140nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485491(CHEMBL2063088)
Affinity DataKi:  2.40nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485494(CHEMBL2063089)
Affinity DataKi:  2.90nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485492(Grazoprevir | Grazoprevir monohydrate | MK-5172 | ...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485494(CHEMBL2063089)
Affinity DataKi:  5.70nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485491(CHEMBL2063088)
Affinity DataKi:  11nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485490(CHEMBL2063087)
Affinity DataKi:  12nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485492(Grazoprevir | Grazoprevir monohydrate | MK-5172 | ...)
Affinity DataKi:  12nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485495(CHEMBL2063085)
Affinity DataKi:  18nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326055((1R,21S,24S)-21-tert-Butyl-N-((1R,2R)-1-{[(cyclopr...)
Affinity DataKi:  22nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485489(CHEMBL1672609 | MK-1220)
Affinity DataKi:  27nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485493(CHEMBL2063086)
Affinity DataKi:  27nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485490(CHEMBL2063087)
Affinity DataKi:  64nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326055((1R,21S,24S)-21-tert-Butyl-N-((1R,2R)-1-{[(cyclopr...)
Affinity DataKi:  77nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485495(CHEMBL2063085)
Affinity DataKi:  79nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485493(CHEMBL2063086)
Affinity DataKi:  80nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50326055((1R,21S,24S)-21-tert-Butyl-N-((1R,2R)-1-{[(cyclopr...)
Affinity DataKi:  88nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485489(CHEMBL1672609 | MK-1220)
Affinity DataKi:  540nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50485489(CHEMBL1672609 | MK-1220)
Affinity DataKi:  790nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332663(CHEMBL1632426)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332664(CHEMBL1632427)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332665(CHEMBL1632428)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332666(CHEMBL1632429)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332667(CHEMBL1632430)
Affinity DataEC50:  3.10E+4nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332668(CHEMBL1632431)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332669(CHEMBL1632432)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332670(CHEMBL1632433)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332671(CHEMBL1632434)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332672(CHEMBL1632435)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332673(CHEMBL1632436)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332674(CHEMBL1632437)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332675(CHEMBL1632438)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332676(CHEMBL1632439)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332677(CHEMBL1632440)
Affinity DataEC50:  2.40E+3nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332678(CHEMBL1632441)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332679(CHEMBL1630184)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332680(CHEMBL1630180)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332681(CHEMBL1630181)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332682(CHEMBL1630182)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332683(CHEMBL1630183)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332684(CHEMBL1630185)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332685(CHEMBL1630186)
Affinity DataEC50:  9.50E+3nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332686(CHEMBL1630187)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332687(CHEMBL1630188)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332688(CHEMBL1630189)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332689(CHEMBL1630190)
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332690(CHEMBL1630191)
Affinity DataEC50:  700nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332691(CHEMBL1630192)
Affinity DataEC50:  700nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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