Affinity DataKi: 0.0500nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease D168V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156T mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Inhibition of Hepatitis C virus (isolate BK) genotype 1b NS3/4a protease A156V mutant expressed in Escherichia coli by time-resolved fluorescence ana...More data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 3.10E+4nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 9.50E+3nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair
TargetPhospholipid-transporting ATPase ABCA1(Mus musculus)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Induction of ABCA1-mediated [3H]cholesterol efflux in mouse J774 macrophages after 4 hrsMore data for this Ligand-Target Pair