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Found 214 with Last Name = 'cil' and Initial = 'o'
TargetBcl-2-like protein 1(Homo sapiens (Human))
Universite De Lyon

Curated by ChEMBL
LigandPNGBDBM50196032((N-[(2-tert-butylbenzenesulfonyl)phenyl]-2,3,4-tri...)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl-xL by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCreatine kinase M-type(Oryctolagus cuniculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50370908(CHEMBL373782)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of rabbit muscle creatine kinase by pH-stat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCreatine kinase M-type(Oryctolagus cuniculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50370908(CHEMBL373782)
Affinity DataKi:  7.00E+4nMAssay Description:Inhibition of rabbit muscle creatine kinase-MgATP complex by pH-stat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519196(CHEMBL4436134)
Affinity DataIC50:  23nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/bicarbonate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519196(CHEMBL4436134)
Affinity DataIC50:  25nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of [3H]norepinephrine uptake in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519191(CHEMBL4464849)
Affinity DataIC50:  35nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/bicarbonate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519191(CHEMBL4464849)
Affinity DataIC50:  40nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519198(CHEMBL4469522)
Affinity DataIC50:  60nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519207(CHEMBL4442662)
Affinity DataIC50:  70nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50:  77nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 20 mins followed by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239467(CHEMBL4086165)
Affinity DataIC50:  80nMAssay Description:Inhibition of TMEM16A (unknown origin) expressed in Xenopus laevis oocytes at -60 mV holding potential by voltage-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50:  83nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519172(CHEMBL4562582)
Affinity DataIC50:  100nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50:  110nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239433(CHEMBL3134585)
Affinity DataIC50:  130nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575379(CHEMBL4852814)
Affinity DataIC50:  150nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239428(CHEMBL4104024)
Affinity DataIC50:  150nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519206(CHEMBL4544784)
Affinity DataIC50:  150nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239446(CHEMBL4069503)
Affinity DataIC50:  170nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239457(CHEMBL4071143)
Affinity DataIC50:  180nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575376(CHEMBL4854119)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239447(CHEMBL4090522)
Affinity DataIC50:  220nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239461(CHEMBL4074900)
Affinity DataIC50:  230nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239457(CHEMBL4071143)
Affinity DataIC50:  230nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239470(CHEMBL4095338)
Affinity DataIC50:  230nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239426(CHEMBL1444023)
Affinity DataIC50:  260nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575384(CHEMBL4866473)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239433(CHEMBL3134585)
Affinity DataIC50:  300nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519171(CHEMBL4457710)
Affinity DataIC50:  300nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575413(CHEMBL4877679)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519185(CHEMBL4445315)
Affinity DataIC50:  300nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239438(CHEMBL4099581)
Affinity DataIC50:  320nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 from rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239475(CHEMBL4082703)
Affinity DataIC50:  370nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239469(CHEMBL4091961)
Affinity DataIC50:  370nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239458(CHEMBL4095365)
Affinity DataIC50:  380nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575404(CHEMBL4863558)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575409(CHEMBL4863725)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-2(Homo sapiens)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239457(CHEMBL4071143)
Affinity DataIC50:  400nMAssay Description:Inhibition of human TMEM16B expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-2(Homo sapiens)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of [3H]5-HT transporter uptake in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575378(CHEMBL4849241)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239426(CHEMBL1444023)
Affinity DataIC50:  420nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239463(CHEMBL4087641)
Affinity DataIC50:  450nMAssay Description:In vitro inhibition of [3H]dopamine uptake in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519203(CHEMBL4550735)
Affinity DataIC50:  450nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239448(CHEMBL4080209)
Affinity DataIC50:  490nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575377(CHEMBL4874714)
Affinity DataIC50:  500nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575383(CHEMBL4849781)
Affinity DataIC50:  500nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519195(CHEMBL4469915)
Affinity DataIC50:  500nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50575387(CHEMBL4848036)
Affinity DataIC50:  500nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChloride anion exchanger(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50519173(CHEMBL4573104)
Affinity DataIC50:  500nMAssay Description:Inhibition of mouse slc26a3 expressed in FRT cells co-expressing EYFP-H148Q/I152L/F46L assessed as reduction in protein-mediated chloride/iodide exch...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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