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Found 8 with Last Name = 'clement' and Initial = 'ja'
TargetTranscription factor Jun(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50295171(AILANTHINONE | CHEMBL487194)
Affinity DataIC50:  32nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50349194(GLAUCARUBINONE | NSC-14975)
Affinity DataIC50:  40nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50295170(6R-senecionylchaparrin | CHEMBL564009)
Affinity DataIC50:  71nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50273917(CHEMBL462089 | Isolissoclinotoxin B)
Affinity DataIC50:  5.86E+4nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50273972(CHEMBL461462 | Lissoclinidine B)
Affinity DataIC50:  5.86E+4nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50273919(CHEMBL513108 | Diplamine B)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50273918(CHEMBL462090 | N,N-dimethyl-5-methylvaracin)
Affinity DataIC50:  1.21E+5nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50240848(2-(3,4-Dimethoxy-5,6,7,8,9-pentathia-benzocyclohep...)
Affinity DataIC50: >2.95E+5nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed