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Found 105 with Last Name = 'cohen' and Initial = 'jh'
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287969((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083490((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083469((R)-3-(5-Chloro-thiophen-2-yl)-3-{[(R)-1-(3-piperi...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287978((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083492((S)-3-(6-Methyl-pyridin-3-yl)-3-{[(R)-1-(3-piperid...)
Affinity DataIC50:  0.130nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083453((S)-3-(6-Chloro-pyridin-3-yl)-3-{[(R)-1-(3-piperid...)
Affinity DataIC50:  0.140nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083456((S)-3-(5-Bromo-pyridin-3-yl)-3-{[(R)-1-(3-piperidi...)
Affinity DataIC50:  0.210nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083479((R)-5-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50:  0.220nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083455((S)-3-(5-Ethynyl-pyridin-3-yl)-3-{[(R)-1-(3-piperi...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083496((R)-3-Benzo[1,3]dioxol-5-yl-3-({(R)-1-[3-(1-methyl...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083467((S)-5-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50:  0.290nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083495((S)-3-(5,6-Dichloro-pyridin-3-yl)-3-{[(R)-1-(3-pip...)
Affinity DataIC50:  0.340nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083478((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.360nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083466((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083471((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083466((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083449((R)-4-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287967((S)-3-Benzo[1,3]dioxol-5-yl-3-{[(R)-1-(3-piperidin...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083482((R)-3-Benzo[1,3]dioxol-5-yl-3-{[(R)-1-(3-piperidin...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083480((S)-3-(5-Phenyl-pyridin-3-yl)-3-{[(R)-1-(3-piperid...)
Affinity DataIC50:  0.520nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083465((S)-3-{[(R)-1-((E)-3-Piperidin-4-yl-acryloyl)-pyrr...)
Affinity DataIC50:  0.580nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083487((S)-3-{[(R)-1-([1,4']Bipiperidinyl-4-carbonyl)-pip...)
Affinity DataIC50:  0.650nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083447((S)-3-(5-Phenethyl-pyridin-3-yl)-3-{[(R)-1-(3-pipe...)
Affinity DataIC50:  0.660nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083448((S)-3-({(R)-1-[3-(1-Iminomethyl-piperidin-4-yl)-pr...)
Affinity DataIC50:  0.75nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083483((S)-3-{[(R)-1-((E)-3-Piperidin-4-yl-acryloyl)-pipe...)
Affinity DataIC50:  0.810nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083475((S)-3-(5-Phenylethynyl-pyridin-3-yl)-3-{[(R)-1-(3-...)
Affinity DataIC50:  0.850nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083462(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083450((S)-3-{[(R)-4-(3-Piperidin-4-yl-propionyl)-piperaz...)
Affinity DataIC50:  1.70nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083488(3-(5-Phenyl-pyridin-3-yl)-3-{[1-(3-piperidin-4-yl-...)
Affinity DataIC50:  1.80nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287983(5-Methyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083460((S)-3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propion...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287982(3-{[1-(3-Piperazin-1-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083494(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083461(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083463((R)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287985(3-Phenyl-3-{[1-(3-piperidin-4-yl-propionyl)-piperi...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287972(2-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083467((S)-5-Phenyl-3-{[(R)-1-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083493(3-(5-Bromo-pyridin-3-yl)-3-{[1-(3-piperidin-4-yl-p...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083459(2-Hydroxy-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-p...)
Affinity DataIC50:  3.5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083489(3-[5-(3-Amino-phenyl)-pyridin-3-yl]-3-{[1-(3-piper...)
Affinity DataIC50:  3.60nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083468((S)-3-(5-Chloro-6-methoxy-pyridin-3-yl)-3-{[(R)-1-...)
Affinity DataIC50:  3.80nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083454((S)-3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperid...)
Affinity DataIC50:  3.80nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287977(3-{[(S)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083452(3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50:  4.80nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083459(2-Hydroxy-3-{[(R)-1-(3-piperidin-4-yl-propionyl)-p...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083476((S)-6,6-Dimethyl-3-{[(R)-1-(3-piperidin-4-yl-propi...)
Affinity DataIC50:  5.60nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobolized fibrinogen receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50083452(3-{[(R)-1-(3-Piperidin-4-yl-propionyl)-piperidine-...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287973(3-({1-[3-(1-Methyl-piperidin-4-yl)-propionyl]-pipe...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50034703(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of biotinylated fibrinogen binding to immobilized integrin alpha IIb beta3More data for this Ligand-Target Pair
In DepthDetails Article
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