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Found 669 with Last Name = 'conner' and Initial = 'se'
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217410(CHEMBL105762)
Affinity DataKi:  0.676nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119704(CHEMBL104809 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217412(CHEMBL322873)
Affinity DataKi:  1.70nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119707(4-[3-(4-Hexanoyl-phenoxy)-propyl]-piperazine-1-car...)
Affinity DataKi:  2nMAssay Description:Binding affinity of the compound towards rats Histamine type 3 (H3) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217416(CHEMBL105515)
Affinity DataKi:  2.10nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119721(CHEMBL103027 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119710(CHEMBL104618 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119735(3-Cyano-N-{(S)-1-[3-(4-cyclopropanecarbonyl-phenox...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50240709((R)-4'-(3-(3-(dimethylamino)pyrrolidin-1-yl)propox...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119722(CHEMBL107162 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119705(CHEMBL101691 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  3nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119712(3-Chloro-N-{(S)-1-[3-(4-cyclopropanecarbonyl-pheno...)
Affinity DataKi:  3nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119701(CHEMBL104808 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119711(2-Chloro-N-{(S)-1-[3-(4-cyclopropanecarbonyl-pheno...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119728(4-Chloro-N-{(S)-1-[3-(4-cyclopropanecarbonyl-pheno...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50404001(CHEMBL2112451)
Affinity DataKi:  4nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217413(CHEMBL2112461)
Affinity DataKi:  4.10nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119720(CHEMBL107293 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119702(CHEMBL102925 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119736(4-Bromo-N-{(S)-1-[3-(4-cyclopropanecarbonyl-phenox...)
Affinity DataKi:  5nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119725(4-tert-Butyl-N-{(S)-1-[3-(4-cyclopropanecarbonyl-p...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119733(CHEMBL102840 | N-{(S)-1-[3-(4-Acetyl-phenoxy)-prop...)
Affinity DataKi:  6nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217096(CHEMBL105267)
Affinity DataKi:  6.20nMAssay Description:Binding affinity at human cloned Histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217410(CHEMBL105762)
Affinity DataKi:  6.5nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217149(CHEMBL102984)
Affinity DataKi:  7.10nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217101(CHEMBL25688)
Affinity DataKi:  7.20nMAssay Description:Binding affinity at human cloned Histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217103(CHEMBL104669)
Affinity DataKi:  8.30nMAssay Description:Binding affinity at human cloned Histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217150(CHEMBL105967)
Affinity DataKi:  8.30nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217408(CHEMBL106545)
Affinity DataKi:  8.5nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217411(CHEMBL323562)
Affinity DataKi:  9.80nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119698(1-Methyl-1H-imidazole-4-sulfonic acid {(S)-1-[3-(4...)
Affinity DataKi:  10nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119730(CHEMBL102929 | N-{(S)-1-[3-(4-Cyclopropanecarbonyl...)
Affinity DataKi:  11nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119708(2-Cyano-N-{(S)-1-[3-(4-cyclopropanecarbonyl-phenox...)
Affinity DataKi:  11nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50240709((R)-4'-(3-(3-(dimethylamino)pyrrolidin-1-yl)propox...)
Affinity DataKi:  13nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217150(CHEMBL105967)
Affinity DataKi:  13nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217411(CHEMBL323562)
Affinity DataKi:  14nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217418(CHEMBL421026)
Affinity DataKi:  15nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217413(CHEMBL2112461)
Affinity DataKi:  15nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217416(CHEMBL105515)
Affinity DataKi:  16nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50404002(CHEMBL2112452)
Affinity DataKi:  17nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50119739(CHEMBL102794 | {4-[3-((1S,4S)-5-Benzenesulfonyl-2,...)
Affinity DataKi:  19nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217102(CHEMBL318801)
Affinity DataKi:  19nMAssay Description:Binding affinity at human cloned Histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217149(CHEMBL102984)
Affinity DataKi:  23nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217099(CHEMBL106483)
Affinity DataKi:  25nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217412(CHEMBL322873)
Affinity DataKi:  26nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217105(CHEMBL320178)
Affinity DataKi:  28nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217415(CHEMBL105669)
Affinity DataKi:  28nMAssay Description:Binding affinity of human cortical histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217408(CHEMBL106545)
Affinity DataKi:  30nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217330(CHEMBL106596)
Affinity DataKi:  30nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50217414(CHEMBL102416)
Affinity DataKi:  32nMAssay Description:Binding affinity at rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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