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Found 13 with Last Name = 'contoreggi' and Initial = 'c'
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087556((4-Fluoro-butyl)-propyl-[2,5,6-trimethyl-7-(2,4,6-...)
Affinity DataKi:  0.910nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  1nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50131716(CHEMBL430892 | [3-(4-Bromo-2-chloro-phenyl)-2,5-di...)
Affinity DataKi:  1.90nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087559(CHEMBL164206 | Cyclopropylmethyl-propyl-[2,5,6-tri...)
Affinity DataKi:  2.30nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  2.5nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50096721(5-Chloro-N-cyclopropylmethyl-N'-(2,6-dichloro-4-tr...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087560(CHEMBL348967 | Ethyl-(4-fluoro-butyl)-[2,5,6-trime...)
Affinity DataKi:  3.5nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087561(Butyl-(4-fluoro-butyl)-[2,5,6-trimethyl-7-(2,4,6-t...)
Affinity DataKi:  10nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50096722(5-Chloro-N-cyclopropylmethyl-N'-(2,6-dichloro-4-io...)
Affinity DataKi:  14nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50096723(CHEMBL113333 | N-(4-Bromo-2,6-dichloro-phenyl)-5-c...)
Affinity DataKi:  21nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087557(CHEMBL164042 | Cyclopropylmethyl-(3-fluoro-propyl)...)
Affinity DataKi:  30nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50054245(5-Chloro-N-cyclopropylmethyl-2-methyl-N-propyl-N''...)
Affinity DataKi:  31nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087558(4-[4-(2-Fluoro-ethyl)-piperazin-1-yl]-2,5,6-trimet...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed