Affinity DataKi: 0.407nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.562nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for 5-hydroxytryptamine 1F receptor was determinedMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation co...More data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity for 5-hydroxytryptamine 1E receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity for Dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP55,940 from human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity for Dopamine receptor D2 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor was determinedMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity for 5-hydroxytryptamine 2B receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inverse agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 7 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of [125I]-MCP-1 binding to the cloned C-C chemokine receptor type 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity of the compound for C-C chemokine receptor type 2B was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair