TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens
Curated by ChEMBL
Agricultural University Of Athens
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by 1-chloro-2,4-dinitrobenzene competitive assayMore data for this Ligand-Target Pair
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens
Curated by ChEMBL
Agricultural University Of Athens
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by 1-chloro-2,4-dinitrobenzene competitive assayMore data for this Ligand-Target Pair
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens
Curated by ChEMBL
Agricultural University Of Athens
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by 1-chloro-2,4-dinitrobenzene competitive assayMore data for this Ligand-Target Pair
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens
Curated by ChEMBL
Agricultural University Of Athens
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by glutathione competitive assayMore data for this Ligand-Target Pair
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens
Curated by ChEMBL
Agricultural University Of Athens
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by glutathione competitive assayMore data for this Ligand-Target Pair
TargetGlutathione S-transferase A1(Homo sapiens (Human))
Agricultural University Of Athens
Curated by ChEMBL
Agricultural University Of Athens
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Inhibition of human GSTA1-1 expressed in Escherichia coli BL21 (DE3) by glutathione competitive assayMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST1 receptor expressed in CHO cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.94nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST4 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST2 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
TargetNeuromedin-B receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 11.2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST1 receptor expressed in CHO cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST1 receptor expressed in CHO cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST3 receptor expressed in Chinese hamster CCL-39 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-[LTT]-SS28 from human SST5 receptor expressed in HEK293 cells after 2 hrs by autoradiographic analysisMore data for this Ligand-Target Pair