TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 692nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 741nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.51E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.78E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.82E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.86E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.04E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.69E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 3.24E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 4.17E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 4.57E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 5.13E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 5.13E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 5.89E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 7.24E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 7.59E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 7.94E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 8.51E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 8.91E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 9.55E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 9.55E+3nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.26E+4nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 1.38E+4nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.29E+4nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 2.45E+4nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 3.09E+4nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universidad De Chile
Curated by ChEMBL
Universidad De Chile
Curated by ChEMBL
Affinity DataKi: 3.24E+4nMAssay Description:Displacement of [3H]diltiazem from benzodiazepine binding site of L-type calcium channel in Wistar rat cerebral cortex membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human PDGFRbeta by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human CDK1 by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human Src kinase by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human AurA kinase by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human Akt1 by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of human ROCK1 by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of EGFR (unknown origin) using omnia tyr peptide 7 substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human MEK1 by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of human FAK by kinase inhibition assayMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human RAF1 by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human ERK1 by kinase inhibition assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human KDR incubated for 50 mins by omnia tyr peptide 8 substrate based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.72E+3nMAssay Description:Inhibition of EGFR (unknown origin) using omnia tyr peptide 7 substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human KDR incubated for 50 mins by omnia tyr peptide 8 substrate based fluorescence assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of human KDR incubated for 50 mins by omnia tyr peptide 8 substrate based fluorescence assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of human KDR incubated for 50 mins by omnia tyr peptide 8 substrate based fluorescence assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of human KDR incubated for 50 mins by omnia tyr peptide 8 substrate based fluorescence assayMore data for this Ligand-Target Pair