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Found 32 with Last Name = 'dagnino' and Initial = 'r'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054245(5-Chloro-N-cyclopropylmethyl-2-methyl-N-propyl-N''...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054252(5-Bromo-N-cyclopropylmethyl-2-methyl-N-propyl-N'-(...)
Affinity DataKi:  2nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054250(CHEMBL306482 | N-Cyclopropylmethyl-2,5-dimethyl-N-...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054248(2,5-Dimethyl-N,N-dipropyl-N'-(2,4,6-trichloro-phen...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054253(CHEMBL77716 | N-Cyclopropylmethyl-5-ethyl-2-methyl...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107083(CHEMBL110609 | [5-(2,4-Dichloro-phenyl)-1-methyl-1...)
Affinity DataKi:  9nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107086(CHEMBL108673 | [5-(4-Bromo-2-methyl-phenyl)-1-meth...)
Affinity DataKi:  10nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107078(2-[5-(2,4-Dichloro-phenyl)-3-dipropylamino-[1,2,4]...)
Affinity DataKi:  14nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107085(CHEMBL323437 | [5-(2,4-Dichloro-5-fluoro-phenyl)-1...)
Affinity DataKi:  15nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107074(CHEMBL106675 | [5-(4-Chloro-2-methyl-phenyl)-1-met...)
Affinity DataKi:  22nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107069(CHEMBL107786 | [5-(4-Chloro-2-methoxy-phenyl)-1-me...)
Affinity DataKi:  26nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054246(CHEMBL77006 | N-Cyclopropylmethyl-2-methyl-N-propy...)
Affinity DataKi:  30nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107080(CHEMBL106728 | [5-(4-Chloro-phenyl)-1-methyl-1H-[1...)
Affinity DataKi:  33nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054225(CHEMBL306618 | N-Cyclopropylmethyl-6-methyl-N-prop...)
Affinity DataKi:  57nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054249(CHEMBL140175 | N*4*-Cyclopropylmethyl-6-methyl-N*4...)
Affinity DataKi:  70nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107076(CHEMBL323257 | Dicyclopropylmethyl-[5-(2,4-dimethy...)
Affinity DataKi:  72nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107084(CHEMBL106972 | [5-(2,4-Dichloro-phenyl)-1-ethyl-1H...)
Affinity DataKi:  80nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107071(CHEMBL110222 | Dicyclopropylmethyl-[1-methyl-5-(2,...)
Affinity DataKi:  120nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054247(CHEMBL344805 | N-Cyclopropylmethyl-2,5,N'-trimethy...)
Affinity DataKi:  150nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054244(CHEMBL134475 | N-Cyclopropylmethyl-2-methyl-N-prop...)
Affinity DataKi:  253nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107072(CHEMBL321155 | Dicyclopropylmethyl-[1-ethyl-5-(2,4...)
Affinity DataKi:  310nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054255(CHEMBL80806 | N-Cyclopropylmethyl-2-methyl-N-propy...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107081(CHEMBL106093 | Dicyclopropylmethyl-propyl-[1-(2,2,...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107070(CHEMBL107091 | [1-Allyl-5-(2,4,6-trimethyl-phenyl)...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107075(CHEMBL175536 | [5-(2,4-Dichloro-phenyl)-1H-[1,2,4]...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107079(CHEMBL431067 | [5-(2,4-Dichloro-phenyl)-1-methyl-1...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107068(CHEMBL108784 | Dicyclopropylmethyl-propyl-[5-(2,4,...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107073(CHEMBL106874 | [5-(2,4-Dichloro-phenyl)-1-methyl-1...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107082(CHEMBL321389 | [5-(2,4-Dichloro-phenyl)-2-methyl-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50107077(CHEMBL110231 | Cyclopropylmethyl-[5-(2,4-dichloro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]-o-CRF binding to human Corticotrophin releasing factor receptor 1 expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054254(CHEMBL136593 | N-Cyclopropylmethyl-N-propyl-N'-(2,...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054251(CHEMBL138687 | N*2*-Cyclopropylmethyl-6-methyl-N*2...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed