Found 158 with Last Name = 'dai' and Initial = 'z' 
Affinity DataIC50: 0nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 0.400nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in mouse BMDMsMore data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Inhibition of NLRP3 in human monocyte-derived macrophagesMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam and testosterone as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS...More data for this Ligand-Target Pair
Affinity DataIC50: 10.2nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 31.7nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 37.6nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 41.1nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 45.5nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 61.2nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 86nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Key Laboratory Of Industrial Fermentation Microbiology (Tianjin University Of Science & Technology)
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-trifluoromethylcoumarin as substrate incubated for 30 mins by fluorescence microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 125nMpH: 7.4Assay Description:Test method: wetting membranes by saponin solution, and preparing [35S]-GTPγS in binding solution (4×). The test compound was prepared as 4× of ...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using paclitaxel as substrate incubated for 5 to 45 mins in presence of NADPH by LC/MS analysisMore data for this Ligand-Target Pair
