Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Leukotriene D4 induced contraction of guinea-pig trachea was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration of the compound against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined (Experiment 2)More data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 2More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determined; experiment 1More data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against [3H]-Leukotriene D4 binding to guinea-pig lung membranes was determinedMore data for this Ligand-Target Pair
TargetP2Y purinoceptor 14(Mus musculus)
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Merck Frosst Center For Therapeutic Research
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Antagonist activity at mouse P2Y14 expressed in human HEK cells coexpressing Galphai5 assessed as inhibition of UDP-glucose stimulated calcium releas...More data for this Ligand-Target Pair