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maximum 50k data
Found 30 with Last Name = 'delcros' and Initial = 'jg'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50069792((2S)-2-[(2S)-2-acetamido-4-methylpentanamido]-N-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475621(CHEMBL371434)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475612(CHEMBL201169)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475614(CHEMBL201249)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475620(CHEMBL372819)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475624(CHEMBL202832)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475615(CHEMBL425927)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475617(CHEMBL433988)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475616(CHEMBL199878)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM86164(N1-DnsSpm | N1-dansyl-spermidine)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of calmodulin dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475623(CHEMBL382499)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475613(CHEMBL102072)
Affinity DataIC50:  1.16E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50216731(CHEMBL158848)
Affinity DataIC50:  1.49E+5nMAssay Description:Inhibition of calmodulin dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50216732(CHEMBL423054)
Affinity DataIC50:  3.13E+5nMAssay Description:Inhibition of calmodulin dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475618(CHEMBL199956)
Affinity DataIC50:  3.73E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475611(CHEMBL275659)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475610(CHEMBL372198)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475609(CHEMBL201076)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475608(CHEMBL383190)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50009385(1,4-butylenediamine | 1,4-tetramethylenediamine | ...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475622(CHEMBL438266)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475619(CHEMBL446186)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50009353(1,5,10-triazadecane | 4-azaoctamethylenediamine | ...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of bovine calmodulin-activated cAMP dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50216729(CHEMBL422519)
Affinity DataIC50:  5.84E+5nMAssay Description:Inhibition of calmodulin dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159158(CHEMBL433563 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159149(CHEMBL179042 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159149(CHEMBL179042 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159158(CHEMBL433563 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50216730(CHEMBL156809)
Affinity DataIC50: >1.50E+6nMAssay Description:Inhibition of calmodulin dependent phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed