Affinity DataKi: 1nM ΔG°: -51.4kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.6kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.6kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.6kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.9kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 15nM ΔG°: -44.7kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 40nM ΔG°: -42.2kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 57nM ΔG°: -41.3kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 73nM ΔG°: -40.7kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 89nM ΔG°: -40.2kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 203nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 206nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 233nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 263nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 264nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 287nM ΔG°: -37.3kJ/molepH: 7.8 T: 2°CAssay Description:The inhibitory effect of test compound for human fXa was determined by using the chromogenic substrates S-2765. The hydrolysis rates of chromogenic s...More data for this Ligand-Target Pair