Compile Data Set for Download or QSAR
maximum 50k data
Found 212 with Last Name = 'filhol' and Initial = 'o'
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)
Affinity DataKi:  180nMAssay Description:Competitive inhibition of recombinant human GST-tagged CK2alpha by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)
Affinity DataKi:  180nMAssay Description:Competitive inhibition of recombinant human GST-tagged CK2alpha by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of N-terminal GST-tagged human CLK2 (138 to end residues) using SR-rich substrate and [gamma-33P]ATP incubated for 40 mins by scintillatio...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of N-terminal GST-tagged human CLK2 (138 to end residues) using SR-rich substrate and [gamma-33P]ATP incubated for 40 mins by scintillatio...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616483(US20230278983, Code AB1455)
Affinity DataIC50:  5.10nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of human recombinant DyrK1b by fluorescence-based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of human recombinant DyrK1b by fluorescence-based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human recombinant DyrK1a by fluorescence-based immunoassayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human recombinant DyrK1a by fluorescence-based immunoassayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616482(US20230278983, Code AB1454)
Affinity DataIC50:  11nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate and [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate and [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616454(US20230278983, Code AB1206)
Affinity DataIC50:  16nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50132260(2-(2-Chloro-4-iodo-phenylamino)-N-cyclopropylmetho...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50132260(2-(2-Chloro-4-iodo-phenylamino)-N-cyclopropylmetho...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616473(US20230278983, Code AB1381)
Affinity DataIC50:  17nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616446(US20230278983, Code AB1073)
Affinity DataIC50:  18nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616474(US20230278983, Code AB1394)
Affinity DataIC50:  23nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616451(US20230278983, Code AB1133)
Affinity DataIC50:  26nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616466(US20230278983, Code AB1303)
Affinity DataIC50:  33nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616423(US20230278983, Code AB668)
Affinity DataIC50:  41nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616481(US20230278983, Code AB1451)
Affinity DataIC50:  45nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616476(US20230278983, Code AB1402)
Affinity DataIC50:  45nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616455(US20230278983, Code AB1208)
Affinity DataIC50:  45nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616449(US20230278983, Code AB1076)
Affinity DataIC50:  46nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616452(US20230278983, Code AB1135)
Affinity DataIC50:  48nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616480(US20230278983, Code AB1450)
Affinity DataIC50:  49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616463(US20230278983, Code AB1287)
Affinity DataIC50:  49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616437(US20230278983, Code AB935 | isobutyl 5-fluoro-3-(1...)
Affinity DataIC50:  49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616450(US20230278983, Code AB1130)
Affinity DataIC50:  49nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616477(US20230278983, Code AB1415)
Affinity DataIC50:  50nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616436(US20230278983, Code AB934)
Affinity DataIC50:  52nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616440(US20230278983, Code AB1030)
Affinity DataIC50:  54nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616432(US20230278983, Code AB929)
Affinity DataIC50:  58nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616435(US20230278983, Code AB933)
Affinity DataIC50:  62nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616444(US20230278983, Code AB1071)
Affinity DataIC50:  65nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616447(US20230278983, Code AB1074)
Affinity DataIC50:  69nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616456(US20230278983, Code AB1209)
Affinity DataIC50:  70nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616429(US20230278983, Code AB914)
Affinity DataIC50:  71nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616434(US20230278983, Code AB932)
Affinity DataIC50:  75nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616464(US20230278983, Code AB1288)
Affinity DataIC50:  78nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616448(US20230278983, Code AB1075)
Affinity DataIC50:  79nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616427(US20230278983, Code AB913)
Affinity DataIC50:  80nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616457(US20230278983, Code AB1210)
Affinity DataIC50:  85nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616459(N-(2-(4-((4-(5-fluoro-2-formyl-1H-indol-3-yl)-1H-1...)
Affinity DataIC50:  90nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616433(US20230278983, Code AB931)
Affinity DataIC50:  100nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616445(US20230278983, Code AB1072)
Affinity DataIC50:  100nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM616478(US20230278983, Code AB1416)
Affinity DataIC50:  100nMAssay Description:All kinase assays were performed as previously described5 at −4° C. in a final volume of 18 μL, containing 2 μL of compounds accordin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 212 total ) | Next | Last >>
Jump to: