Affinity DataKi: 0.530nMAssay Description:Inhibition assay using matrix metalloproteinase (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition assay using matrix metalloproteinase (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:In vitro inhibitory activity against biotinylated human HIV-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of Pseudomonas aeruginosa PAO1 NagZ using PNP-GlcNAc as substrate assessed as release of 4-nitrophenolate ion after 4 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition assay using matrix metalloproteinase (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition assay using matrix metalloproteinase (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition assay using matrix metalloproteinase (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Competitive inhibition of Pseudomonas aeruginosa PAO1 NagZ using PNP-GlcNAc as substrate assessed as release of 4-nitrophenolate ion after 4 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:Competitive inhibition of Pseudomonas aeruginosa PAO1 NagZ using PNP-GlcNAc as substrate assessed as release of 4-nitrophenolate ion after 4 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition assay using matrix metalloproteinase (MMP-2).Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+4nMAssay Description:Competitive inhibition of Pseudomonas aeruginosa PAO1 NagZ using PNP-GlcNAc as substrate assessed as release of 4-nitrophenolate ion after 4 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 49.7nMAssay Description:Binding affinity to methicillin-susceptible Staphylococcus aureus PBP 2More data for this Ligand-Target Pair
TargetPenicillin-binding protein, transpeptidase domain protein(Staphylococcus aureus)
University Of Notre Dame
Curated by ChEMBL
University Of Notre Dame
Curated by ChEMBL
Affinity DataIC50: 71.6nMAssay Description:Binding affinity to methicillin-susceptible Staphylococcus aureus PBP 3More data for this Ligand-Target Pair
TargetPenicillin-binding protein, transpeptidase domain protein(Staphylococcus aureus)
University Of Notre Dame
Curated by ChEMBL
University Of Notre Dame
Curated by ChEMBL
Affinity DataIC50: 72.4nMAssay Description:Inhibition of methicillin-susceptible Staphylococcus aureus ATCC 29213 PBP 3More data for this Ligand-Target Pair
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
University Of Notre Dame
Curated by ChEMBL
University Of Notre Dame
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Inhibition of methicillin-susceptible Staphylococcus aureus ATCC 29213 PBP 1More data for this Ligand-Target Pair
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
University Of Notre Dame
Curated by ChEMBL
University Of Notre Dame
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Binding affinity to methicillin-susceptible Staphylococcus aureus PBP 1More data for this Ligand-Target Pair
Affinity DataIC50: 233nMAssay Description:Inhibition of methicillin-resistant Staphylococcus aureus PBP 2aMore data for this Ligand-Target Pair
Affinity DataIC50: 262nMAssay Description:Binding affinity to methicillin-resistant Staphylococcus aureus MF535HR PBP 2a by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 723nMAssay Description:Inhibition of methicillin-susceptible Staphylococcus aureus ATCC 29213 PBP 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of methicillin-resistant Staphylococcus aureus OC 3726 PBP 2aMore data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of methicillin-susceptible Staphylococcus aureus ATCC 29213 PBP 4More data for this Ligand-Target Pair
Affinity DataIC50: >1.46E+3nMAssay Description:Binding affinity to methicillin-susceptible Staphylococcus aureus PBP 4More data for this Ligand-Target Pair
TargetMembrane-bound lytic murein transglycosylase B(Escherichia coli (strain K12))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKd: 1.01E+6nMAssay Description:Binding affinity to Escherichia coli K12 MG1655 His6x-tagged MltB lytic transglycosylase assessed as intrinsic fluorescence of tryptophan and/or tyro...More data for this Ligand-Target Pair
TargetMembrane-bound lytic murein transglycosylase B(Escherichia coli (strain K12))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKd: 1.00E+6nMAssay Description:Binding affinity to Escherichia coli K12 MG1655 His6x-tagged MltB lytic transglycosylase assessed as intrinsic fluorescence of tryptophan and/or tyro...More data for this Ligand-Target Pair
TargetMembrane-bound lytic murein transglycosylase B(Escherichia coli (strain K12))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKd: 1.89E+5nMAssay Description:Binding affinity to Escherichia coli K12 MG1655 His6x-tagged MltB lytic transglycosylase assessed as intrinsic fluorescence of tryptophan and/or tyro...More data for this Ligand-Target Pair
TargetMembrane-bound lytic murein transglycosylase B(Escherichia coli (strain K12))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKd: 1.74E+5nMAssay Description:Binding affinity to Escherichia coli K12 MG1655 His6x-tagged MltB lytic transglycosylase assessed as intrinsic fluorescence of tryptophan and/or tyro...More data for this Ligand-Target Pair