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maximum 50k data
Found 333 with Last Name = 'forn' and Initial = 'j'
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003524(CHEMBL3216197 | [4-(2,2-Diphenyl-propionyl)-pipera...)
Affinity DataIC50:  1.90nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005224(2-({Acetyl-[5-(16-methoxy-hexadecyloxy)-tetrahydro...)
Affinity DataIC50:  2.10nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003499(CHEMBL338940 | [4-(3-Hydroxy-3,3-diphenyl-propiony...)
Affinity DataIC50:  2.70nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 in U-937 cells from human histiocytic lymphomaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005227(2-({Acetyl-[5-(6-decyloxy-hexyloxy)-tetrahydro-fur...)
Affinity DataIC50:  4.10nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011053(CHEMBL125576 | Tetrahydrofuran derivative)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005225(2-{[Acetyl-(5-hexadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  6.80nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003525(CHEMBL133742 | [4-(2,3-Diphenyl-acryloyl)-piperazi...)
Affinity DataIC50:  7.5nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011106(2-{[Acetyl-(4-octadecyloxymethyl-[1,3]dioxolan-2-y...)
Affinity DataIC50:  7.5nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011053(CHEMBL125576 | Tetrahydrofuran derivative)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011055(2-{[Acetyl-(4-hexadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  8.20nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005225(2-{[Acetyl-(5-hexadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  8.60nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005225(2-{[Acetyl-(5-hexadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  8.60nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045990(CHEMBL102070 | N-(3-{4-[Cyano-(2-methyl-pyridin-3-...)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Prostaglandin G/H synthase 2 in 143.98.2 from human osteosarcoma cellsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045970(CHEMBL102918 | N-(3-{4-[Cyano-(2-methyl-pyridin-3-...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003506(CHEMBL322184 | CHEMBL545771 | {4-[2-(Benzhydryl-am...)
Affinity DataIC50:  9.10nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003506(CHEMBL322184 | CHEMBL545771 | {4-[2-(Benzhydryl-am...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50046012(CHEMBL100497 | [4-(3-Benzylamino-3-phenyl-propiony...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005231(2-{[Acetyl-(5-hexadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  9.70nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003522((4-Diphenylacetyl-piperazin-1-yl)-pyridin-3-yl-ace...)
Affinity DataIC50:  10nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003473(CHEMBL317193 | [4-(3,3-Diphenyl-acryloyl)-piperazi...)
Affinity DataIC50:  10nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003473(CHEMBL317193 | [4-(3,3-Diphenyl-acryloyl)-piperazi...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of PAF-induced platelet aggregation in male rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005237(2-{[Acetyl-(5-octadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011058(CHEMBL124534 | Tetrahydrofuran derivative)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003514(CHEMBL3216401 | [4-(2-Benzyl-3-phenyl-propionyl)-p...)
Affinity DataIC50:  11nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045982(CHEMBL103596 | [4-(3-Methylamino-3-phenyl-propiony...)
Affinity DataIC50:  11nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011058(CHEMBL124534 | Tetrahydrofuran derivative)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045983(CHEMBL103393 | [3-{4-[Cyano-(2-methyl-pyridin-3-yl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50046017((2-Methyl-pyridin-3-yl)-[4-(4,4,4-trifluoro-3-phen...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of PAF-induced platelet aggregation in male rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50102311(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-6...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Prostaglandin G/H synthase 2 in 143.98.2 from human osteosarcoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50102309(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-7...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Prostaglandin G/H synthase 2 in 143.98.2 from human osteosarcoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045959(CHEMBL103476 | {4-[2-(Benzhydryl-amino)-propionyl]...)
Affinity DataIC50:  13nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045993((3-{4-[Cyano-(2-methyl-pyridin-3-yl)-methyl]-piper...)
Affinity DataIC50:  14nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045972((2-Methyl-pyridin-3-yl)-[4-(4,4,4-trifluoro-3-hydr...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of PAF-induced platelet aggregation in male rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011058(CHEMBL124534 | Tetrahydrofuran derivative)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005230(2-[(Acetyl-{5-[6-(biphenyl-4-ylmethoxy)-hexyloxy]-...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005226(2-[(Acetyl-{5-[6-(5-phenyl-pentyloxy)-hexyloxy]-te...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011072(CHEMBL126958 | Dioxolane derivative)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50003503(1-(3,3-Diphenyl-propionyl)-4-(pyridin-3-ylamino)-p...)
Affinity DataIC50:  15nMAssay Description:Concentration tested in vitro to inhibit PAF-induced maximum aggregation (PAF-Antagonistic activity) by 50%.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011109(2-{[Acetyl-(4-hexadecyloxymethyl-[1,3]dioxolan-2-y...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50005235(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045964((3-{4-[Cyano-(2-methyl-pyridin-3-yl)-methyl]-piper...)
Affinity DataIC50:  16nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50045995(CHEMBL100641 | [4-(3-Hydroxy-3,3-diphenyl-propiony...)
Affinity DataIC50:  17nMAssay Description:Inhibition of PAF-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50011055(2-{[Acetyl-(4-hexadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & C£A.S.A.

Curated by ChEMBL
LigandPNGBDBM50046027(CHEMBL103231 | N-(3-{4-[Cyano-(2-methyl-pyridin-3-...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of PAF-induced platelet aggregation in male rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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