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Found 37 with Last Name = 'forster' and Initial = 'pi'
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  5nMAssay Description:Inhibition of glucocorticoid receptor-glucocorticoid complex transfected in rat R1 cells assessed as down-regulation of TPA-responsive element proinf...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]naloxone from kappa opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  138nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarboxypeptidase B(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50233004(2-(3-carbamimidamidopropylidene)butanedioic acid |...)
Affinity DataIC50:  360nMAssay Description:Inhibition of carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316549(CHEMBL1097805 | longanine)
Affinity DataIC50:  700nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50216277(4,4'-((1R,2R,3S,4S)-3,4-dimethylcyclobutane-1,2-di...)
Affinity DataIC50:  900nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50095839(CHEMBL3590599)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Tdp1 (unknown origin) incubated for 30 mins using 5'-/6-TAMN/AGGATCTAAAAGACTT/3BHQ_2/-3' substrate by microplate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50095838(CHEMBL3590600)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Tdp1 (unknown origin) incubated for 30 mins using 5'-/6-TAMN/AGGATCTAAAAGACTT/3BHQ_2/-3' substrate by microplate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269337(CHEMBL497516 | Grandisine F)
Affinity DataIC50:  1.55E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269336(grandisine D)
Affinity DataIC50:  1.65E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316551(CHEMBL1096481 | N-methylstephuline)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316546(CHEMBL1097077 | N-methylstephisoferulin)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316547(6-cinnamoylhernandine | CHEMBL1097804)
Affinity DataIC50:  5.10E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316552(CHEMBL1096482 | prostephabyssine)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269357((-)-isoelaeocarpiline | CHEMBL521711)
Affinity DataIC50:  9.90E+3nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316545(6-cinnamoyl-N-methylstephasunoline | CHEMBL1098354)
Affinity DataIC50:  1.13E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50228176(peripentadenine)
Affinity DataIC50:  1.14E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50216279(CHEMBL388363 | di-O-methylendiandrin A)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269339(CHEMBL509995 | Grandisine C)
Affinity DataIC50:  1.46E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316550(CHEMBL1097185 | aknadilactam)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261174(CHEMBL496930 | corymbone B)
Affinity DataIC50:  1.90E+4nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50072394(1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyr...)
Affinity DataIC50:  2.30E+4nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50261685(CHEMBL447346 | corymbone A)
Affinity DataIC50:  2.30E+4nMAssay Description:Displacement of [3H]3-methylhistidyl-TRH from rat recombinant TRH2 receptor expressed in HEK2935 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50216278(CHEMBL228326 | nectandrin B)
Affinity DataIC50:  2.70E+4nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50228177(peripentonine C)
Affinity DataIC50:  3.09E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50216280(CHEMBL228655 | di-O-acetylendiandrin A)
Affinity DataIC50:  3.40E+4nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50216276((-)-dihydroguaiaretic acid | 4,4'-((2R,3R)-2,3-dim...)
Affinity DataIC50:  3.50E+4nMAssay Description:Binding affinity to glucocorticoid receptor by GR binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50260779(CHEMBL524026 | sinococuline)
Affinity DataIC50:  3.70E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316548(CHEMBL1098359 | aknadinine)
Affinity DataIC50:  4.60E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269338(Grandisine G)
Affinity DataIC50:  7.54E+4nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of glucocorticoid receptor-glucocorticoid complex transfected in rat R1 cells assessed as down-regulation of TPA-responsive element proinf...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of glucocorticoid receptor-glucocorticoid complex transfected in rat R1 cells assessed as down-regulation of TPA-responsive element proinf...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed