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Found 34 with Last Name = 'fröhner' and Initial = 'w'
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353649(CHEMBL1829835)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353651(CHEMBL1829841)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353652(CHEMBL1829842)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353649(CHEMBL1829835)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353651(CHEMBL1829841)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353650(CHEMBL1829837)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353648(CHEMBL1829833)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353655(CHEMBL1829834)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353652(CHEMBL1829842)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353654(CHEMBL1829822)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353654(CHEMBL1829822)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353655(CHEMBL1829834)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353650(CHEMBL1829837)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353648(CHEMBL1829833)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50399645(CHEMBL1213203)
Affinity DataEC50:  1.42E+4nMAssay Description:Increase in thermal stability of PDK1 by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50399648(CHEMBL2177686)
Affinity DataEC50:  3.02E+4nMAssay Description:Increase in thermal stability of PDK1 by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50399647(CHEMBL2177670)
Affinity DataEC50:  6.00E+4nMAssay Description:Increase in thermal stability of PDK1 by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50399646(CHEMBL2177668 | PS210)
Affinity DataEC50:  8.58E+4nMAssay Description:Increase in thermal stability of PDK1 by differential scanning fluorimetryMore data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50399645(CHEMBL1213203)
Affinity DataKd:  43nMAssay Description:Binding affinity to PDK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296956((Z)-5-(1H-Indol-3-yl)-3-phenylpent-2-enoic Acid | ...)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296955((Z)-5-(Naphthalen-2-yl)-3-phenylpent-2-enoic Acid ...)
Affinity DataKd:  1.38E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296954((Z)-5-(4-bromo-2-fluorophenyl)-3-phenylpent-2-enoi...)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296953((Z)-5-(2,4-Dichlorophenyl)-3-phenylpent-2-enoic Ac...)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296952((Z)-5-(3,4-Dichlorophenyl)-3-phenylpent-2-enoic Ac...)
Affinity DataKd:  1.39E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296951((Z)-3-Phenyl-5-(4-(trifluoromethyl)phenyl)pent-2-e...)
Affinity DataKd:  1.04E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50399649(CHEMBL2177659)
Affinity DataEC50:  1.30E+4nMAssay Description:Increase in thermal stability of PDK1 by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296949((2Z)-5-(4-chlorophenyl)-3-phenylpent-2-enoic acid ...)
Affinity DataKd:  1.03E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296950((Z)-5-(4-Bromophenyl)-3-phenylpent-2-enoic acid | ...)
Affinity DataKd:  2.09E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed