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Found 260 with Last Name = 'gagginapally' and Initial = 'sr'
LigandPNGBDBM50403292(CHEMBL5285364)
Affinity DataIC50:  950nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50391288(CHEMBL5288438)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50456116(Prx-03140)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against Dihydrofolate reductase in rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50391287(CHEMBL5278176)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50391258(CHEMBL5286257)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50456121(CHEMBL4205936)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50456112(CHEMBL4215911)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM325596(3-[5-(1-Cyclobutyl-piperidin-4-yl)-[1,3,4]oxadiazo...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391288(CHEMBL5288438)
Affinity DataIC50:  2.80E+3nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50391298(CHEMBL5275605)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM325561(1-Isopropyl-3-{5-[1-(3-methoxy propyl) piperidin-4...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM325602(1-Isopropyl-3-{5-[1-(tetrahydro-pyran-4-ylmethyl)-...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM325561(1-Isopropyl-3-{5-[1-(3-methoxy propyl) piperidin-4...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391267(CHEMBL5289747)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50391246(CHEMBL5275895)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat microsomal HMG-CoA reductase activity by 50%More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50456112(CHEMBL4215911)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate after 12 mins in presence of NADPH-regeneration system by LC-MS/MS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50456121(CHEMBL4205936)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate after 2 mins in presence of NADPH-regeneration system by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50456121(CHEMBL4205936)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate after 12 mins in presence of NADPH-regeneration system by LC-MS/MS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50456112(CHEMBL4215911)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate after 2 mins in presence of NADPH-regeneration system by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50391283(CHEMBL5268064)
Affinity DataIC50: >1.00E+4nMAssay Description:Evaluated for inhibitory activity against rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391281(CHEMBL5286642)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391281(CHEMBL5286642)
Affinity DataIC50:  1.39E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig right atriaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391266(CHEMBL5271080)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391278(CHEMBL5274204)
Affinity DataIC50:  2.67E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM325598(3-[5-(1-Cyclopropylmethyl-piperidin-4-yl)-[1,3,4]o...)
Affinity DataIC50:  3.60E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig left atriaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391265(CHEMBL5276171)
Affinity DataIC50:  3.64E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM325596(3-[5-(1-Cyclobutyl-piperidin-4-yl)-[1,3,4]oxadiazo...)
Affinity DataIC50:  3.70E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig right atriaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50403292(CHEMBL5285364)
Affinity DataIC50:  3.77E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-2 adrenergic receptor from guinea pig trachea.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391298(CHEMBL5275605)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for alpha-adrenergic activity against Alpha-1 adrenergic receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM325602(1-Isopropyl-3-{5-[1-(tetrahydro-pyran-4-ylmethyl)-...)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig left atriaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM325561(1-Isopropyl-3-{5-[1-(3-methoxy propyl) piperidin-4...)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig right atriaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391283(CHEMBL5268064)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig left atriaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM325594(3-[5-(1-Cyclobutylmethyl-piperidin-4-yl)-[1,3,4]ox...)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig left atriaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM325597(1-Isopropyl-3-[5-(1-isopropyl-piperidin-4-yl)-[1,3...)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig right atriaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391278(CHEMBL5274204)
Affinity DataIC50: >4.50E+4nMAssay Description:The compound was tested for beta-adrenergic activity against Beta-1 adrenergic receptor from guinea pig right atriaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391267(CHEMBL5289747)
Affinity DataIC50: >4.50E+4nMAssay Description:Antagonistic activity against Thromboxane A2 receptor in guinea pig trachea in the presence of 11,9-epoxymethano-PGH2More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391266(CHEMBL5271080)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391265(CHEMBL5276171)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391248(CHEMBL5284140)
Affinity DataIC50: >4.50E+4nMAssay Description:Evaluated for inhibitory activity against rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50391246(CHEMBL5275895)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50403292(CHEMBL5285364)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391298(CHEMBL5275605)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391288(CHEMBL5288438)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM325602(1-Isopropyl-3-{5-[1-(tetrahydro-pyran-4-ylmethyl)-...)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391283(CHEMBL5268064)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM325596(3-[5-(1-Cyclobutyl-piperidin-4-yl)-[1,3,4]oxadiazo...)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM325598(3-[5-(1-Cyclopropylmethyl-piperidin-4-yl)-[1,3,4]o...)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM325597(1-Isopropyl-3-[5-(1-isopropyl-piperidin-4-yl)-[1,3...)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391248(CHEMBL5284140)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50391246(CHEMBL5275895)
Affinity DataIC50: >4.50E+4nMAssay Description:Inhibition of rabbit lung angiotensin I converting enzyme (ACE) using hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
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