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Found 188 with Last Name = 'galli' and Initial = 'g'
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200018((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  1nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200018((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200015((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  9.90nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200015((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200020((3S,4S)-4-((2S,3S)-2-(4-(4-((4-(6-methoxyquinolin-...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200017((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-amino-1-...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200019((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200021((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-(1-(4-(6-methoxyqu...)
Affinity DataKi:  12nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200019((S)-2-(2S-(4-(4-(((2S,3S)-1-((3S,4S)-1-(butylamino...)
Affinity DataKi:  17nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200014((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  26nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200017((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-amino-1-...)
Affinity DataKi:  33nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200023((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  58nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50146527((3S,4S)-N-butyl-3-hydroxy-6-methyl-4-((2S,3S)-3-me...)
Affinity DataKi:  59nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200014((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  74nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200020((3S,4S)-4-((2S,3S)-2-(4-(4-((4-(6-methoxyquinolin-...)
Affinity DataKi:  81nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200023((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(1-(4-(6-me...)
Affinity DataKi:  103nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50146524((S)-3-(S)-Hydroxy-4-{(S)-3-methyl-2-[2-(naphthalen...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50223627(CHEMBL3215350)
Affinity DataKi:  180nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200016((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-(tert-bu...)
Affinity DataKi:  230nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200016((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-((S)-1-(6-(tert-bu...)
Affinity DataKi:  403nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50146527((3S,4S)-N-butyl-3-hydroxy-6-methyl-4-((2S,3S)-3-me...)
Affinity DataKi:  727nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50200021((3S,4S)-4-((2S,3S)-2-(4-(4-((S)-(1-(4-(6-methoxyqu...)
Affinity DataKi:  765nMAssay Description:Inhibition of Plasmodium falciparum recombinant PLM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50366912(CHEMBL1790774)
Affinity DataIC50:  0.590nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50366909(CHEMBL1790773)
Affinity DataIC50:  1.5nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50366908(CHEMBL1790772)
Affinity DataIC50:  9.60nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587363(CHEMBL5081562)
Affinity DataIC50:  23nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50272529(3,7-Bis(2-hydroxyethyl)icaritin | CHEMBL498486)
Affinity DataIC50:  74nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50146530((S)-2-[4-(4-{(S)-1-[(S)-1-((S)-2-Butylcarbamoyl-1-...)
Affinity DataIC50:  123nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50366910(CHEMBL1790776)
Affinity DataIC50:  135nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50272526(CHEMBL497293 | Icariside II)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha'(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human PDE6CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50272528(7-(2-Hydroxyethyl)-3-O-rhamnosylicariin | CHEMBL50...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50366911(CHEMBL1790775)
Affinity DataIC50:  396nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50240974(2-(3,4-Dihydroxy-phenyl)-3,5,7-trihydroxy-8-(3-met...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50146528(6-Amino-2-(S)-amino-hexanoic acid [4-(6-methoxy-qu...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50240972(5,7-Dihydroxy-2-(4-hydroxy-phenyl)-8-(3-methyl-but...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Milan-Bicocca

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50272527(3-hydroxy-7-o-beta-glucose-8-prenyl-4'-methoxy Chr...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587444(CHEMBL5090997)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587444(CHEMBL5090997)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Milan-Bicocca

Curated by ChEMBL
LigandPNGBDBM50485110(CHEMBL2032213)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Milan-Bicocca

Curated by ChEMBL
LigandPNGBDBM50485110(CHEMBL2032213)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Milan-Bicocca

Curated by ChEMBL
LigandPNGBDBM50485109(CHEMBL2032319)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Milan-Bicocca

Curated by ChEMBL
LigandPNGBDBM50485109(CHEMBL2032319)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587409(CHEMBL5094784)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587409(CHEMBL5094784)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
University Of Milan

Curated by ChEMBL
LigandPNGBDBM50027363(CHEBI:78420 | Icariin)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human recombinant PDE5A1 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587406(CHEMBL5071769)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGTPase KRas(Homo sapiens (Human))
Cambridge University

Curated by ChEMBL
LigandPNGBDBM50587406(CHEMBL5071769)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of alexa fluor 647-labeled kinase tracer 314 binding to biotinylated-KRAS G12V mutant (unknown origin) measured after 60 mins by HTRF comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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