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Found 176 with Last Name = 'gandhi' and Initial = 's'
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin) after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of CDK1/cyclin E (unknown origin) after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263041(CHEMBL4103469)
Affinity DataIC50:  12nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) using histone H1 as substrate after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM24226(1-[(4-fluorophenyl)methyl]-N-{1-[2-(4-methoxypheny...)
Affinity DataIC50:  14nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using YSPTSPSYSPTSPSYSPTSPKKK as substrate after 30 mins in presence of [33P]-gamma-ATP by filter bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  16nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) using histone H1 as substrate after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  16nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using YSPTSPSYSPTSPSYSPTSPKKK as substrate after 30 mins in presence of [33P]-gamma-ATP by filter bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  16nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using YSPTSPSYSPTSPSYSPTSPKKK as substrate after 30 mins in presence of [33P]-gamma-ATP by filter bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50193086(CHEMBL3969723)
Affinity DataIC50:  20nMAssay Description:Inhibition of human SPPL2a expressed in human U2OS cells using EGFP-labeled TNFalpha (1 to 76 residues) NTF as substrate after 24 hrs by Hoechst stai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using YSPTSPSYSPTSPSYSPTSPKKK as substrate after 30 mins in presence of [33P]-gamma-ATP by filter bindi...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  23nMAssay Description:Inhibition of full length recombinant C-terminal 6His-tagged human Cdk9/full-length human Cyclin T1 after 60 mins in presence of [33P]-gamma-ATP by f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263027(CHEMBL4066369)
Affinity DataIC50:  29nMAssay Description:Inhibition of CDK3/cyclin E (unknown origin) after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204980((E)-2-(5-((2-acetamidothiazol-4-yl)methyl)-4-(4-ch...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204969(2-(5-((2-benzamidothiazol-4-yl)methyl)-4-(4-chloro...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205012((E)-N'-benzylidene-2-(5-((2-(2-chloroacetamido)thi...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204973(2-(5-((2-(2-chloroacetamido)thiazol-4-yl)methyl)-4...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  45nMAssay Description:Inhibition of CDK5/cyclin p35 (unknown origin) after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204959(CHEMBL390918 | N-{4-[(4-amino-5-sulfanyl-4H-1,2,4-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1/G1/S-specific cyclin-E2(Homo sapiens (Human))
Dr. Reddys Laboratories

Curated by ChEMBL
LigandPNGBDBM50204959(CHEMBL390918 | N-{4-[(4-amino-5-sulfanyl-4H-1,2,4-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human cdk2/cyclin E by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1/G1/S-specific cyclin-E2(Homo sapiens (Human))
Dr. Reddys Laboratories

Curated by ChEMBL
LigandPNGBDBM50205012((E)-N'-benzylidene-2-(5-((2-(2-chloroacetamido)thi...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human cdk2/cyclin E by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205002(CHEMBL399828 | N-(3-((2-acetamidothiazol-4-yl)meth...)
Affinity DataIC50:  62nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50193086(CHEMBL3969723)
Affinity DataIC50:  63nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) using histone H1 as substrate after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205055(3-{4-[4-(4-chloro-benzoylamino)-5-hydrazinocarbony...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205021(CHEMBL437560 | N-[3-(2-benzoylamino-thiazol-4-ylme...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263011(CHEMBL4100359)
Affinity DataIC50:  66nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using YSPTSPSYSPTSPSYSPTSPKKK as substrate after 30 mins in presence of [33P]-gamma-ATP by filter bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204957(2-(5-((2-acetamidothiazol-4-yl)methyl)-4-(4-chloro...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G1/S-specific cyclin- 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  76nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-O/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  138nMAssay Description:Inhibition of CDK2/cyclin O (unknown origin) after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263045(CHEMBL4074270)
Affinity DataIC50:  160nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) using histone H1 as substrate after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205023(3-{4-[5-[5-[2-(2-carboxy-ethylamino)-thiazol-4-ylm...)
Affinity DataIC50:  168nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205067(3-{4-[5-{2-[N'-(2-chloro-acetyl)-hydrazino]-2-oxo-...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205009(CHEMBL233519 | N-[3-(2-benzoylamino-thiazol-4-ylme...)
Affinity DataIC50:  186nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205016(2-(4-acetamido-5-((2-benzamidothiazol-4-yl)methyl)...)
Affinity DataIC50:  186nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205059(2-(5-((2-acetamidothiazol-4-yl)methyl)-4-benzamido...)
Affinity DataIC50:  197nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263013(CHEMBL4079206)
Affinity DataIC50:  199nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using YSPTSPSYSPTSPSYSPTSPKKK as substrate after 30 mins in presence of [33P]-gamma-ATP by filter bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205035(2-(4-acetamido-5-((2-(2-chloroacetamido)thiazol-4-...)
Affinity DataIC50:  201nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204999(4-chloro-N-(3-[2-(2-chloro-acetylamino)-thiazol-4-...)
Affinity DataIC50:  224nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205049(3-(4-{4-(4-chloro-benzoylamino)-5-[1-phenyl-meth-(...)
Affinity DataIC50:  238nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205033(2-(4-acetamido-5-((2-acetamidothiazol-4-yl)methyl)...)
Affinity DataIC50:  241nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204995(2-(4-benzamido-5-((2-(2-chloroacetamido)thiazol-4-...)
Affinity DataIC50:  246nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205061((E)-2-(5-((2-benzamidothiazol-4-yl)methyl)-4-(4-ch...)
Affinity DataIC50:  246nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263030(CHEMBL4094775)
Affinity DataIC50:  260nMAssay Description:Inhibition of SPPL2a in mouse whole blood assessed as increase in CD74/p8 accumulation after 5.5 hrs by Western bot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204998(CHEMBL232077 | N-(3-(2-acetylamino-thiazol-4-ylmet...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204996(3-[4-(4-acetylamino-5-{2-[N'-(2-chloro-acetyl)-hyd...)
Affinity DataIC50:  264nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205052(3-{N-(4-[(4-amino-5-sulfanyl-4H-1,2,4-triazol-3-yl...)
Affinity DataIC50:  264nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204972(2-(4-benzamido-5-((2-benzamidothiazol-4-yl)methyl)...)
Affinity DataIC50:  268nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50204974(3-{4-[5-[2-(N'-benzoyl-hydrazino)-2-oxo-ethylsulfa...)
Affinity DataIC50:  268nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50263012(CHEMBL4065874)
Affinity DataIC50:  280nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) using histone H1 as substrate after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50205039(CHEMBL399387 | methyl 2-(5-((2-benzamidothiazol-4-...)
Affinity DataIC50:  290nMAssay Description:Inhibition of human cdk5/p25 by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50189885(Rohitukine)
Affinity DataIC50:  300nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) using histone H1 as substrate after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Csir-Indian Institute of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50189885(Rohitukine)
Affinity DataIC50:  300nMAssay Description:Inhibition of human Cdk9/T1 using YSPTSPSYSPTSPSYSPTSPKKK peptide as substrate after 30 mins by 33P-ATP filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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