TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat heartMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 4.96E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II); Range = 32-235 microMMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 3.05E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
Affinity DataIC50: 4.75E+5nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT)More data for this Ligand-Target Pair
Affinity DataIC50: 9.12E+5nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT)More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+6nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT); Range = 1300-4000 microMMore data for this Ligand-Target Pair
Affinity DataKd: 7.70E+3nMAssay Description:Binding affinity to LANCL2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair