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Found 21 with Last Name = 'gandour' and Initial = 'rd'
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataKi:  2.80E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataKi:  4.20E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230709(CHEMBL295954)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230703(CHEMBL296591)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230702(CHEMBL48695)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230712(CHEMBL52232)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230714(CHEMBL48551)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230705(CHEMBL49951)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230711(CHEMBL441041)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230704(CHEMBL416830)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230713(CHEMBL301124)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230701(CHEBI:73067 | Palmitoyl-carnitine)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataIC50:  4.96E+4nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50230710(CHEMBL49275)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of protein kinase C (PKC) purified from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284164((S)-2-Hexadecyl-2-hydroxy-4,4-dimethyl-morpholin-4...)
Affinity DataIC50:  2.35E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II); Range = 32-235 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Louisiana State University

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  3.05E+5nMAssay Description:Inhibitory potency of the compound against Carnitine Palmitoyltransferase (CPT-II)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal carnitine O-octanoyltransferase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  4.75E+5nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal carnitine O-octanoyltransferase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284163((S)-4-Hexadecyl-2,6,6-trimethyl-2-oxo-2lambda*5*-[...)
Affinity DataIC50:  9.12E+5nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisomal carnitine O-octanoyltransferase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284164((S)-2-Hexadecyl-2-hydroxy-4,4-dimethyl-morpholin-4...)
Affinity DataIC50:  4.00E+6nMAssay Description:Inhibitory potency of the compound against carnitine octanoyltransferase (COT); Range = 1300-4000 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLanC-like protein 2(Homo sapiens (Human))
Biotherapeutics

Curated by ChEMBL
LigandPNGBDBM50558735(CHEMBL4788758)
Affinity DataKd:  7.70E+3nMAssay Description:Binding affinity to LANCL2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed