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Found 44 with Last Name = 'garcia' and Initial = 'ga'
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125769(2,6-Diamino-8-phenylsulfanylmethyl-3H-quinazolin-4...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125773(2-Amino-6-methyl-3H-pteridin-4-one | CHEMBL14913)
Affinity DataKi:  250nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125771(6-Amino-2,3-dihydro-benzo[g]phthalazine-1,4-dione ...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125772(2-amino-4-hydroxypteridine | 2-aminopteridin-4-ol ...)
Affinity DataKi:  600nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125760(2-Amino-8-(4-chloro-benzylsulfanyl)-1,9-dihydro-pu...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125766(2-Amino-7-phenyl-3H-pteridin-4-one | CHEMBL277561)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125761(3-Methyl-6,7-dihydro-4H-1-thia-4,6,7-triaza-cyclop...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125768(6,7-Dihydro-4H-1-thia-4,6,7-triaza-cyclopenta[b]na...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125765(3-Amino-6-hydroxy-2-(2-hydroxy-ethyl)-2,5-dihydro-...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125767(4-AMINOPHTHALHYDRAZIDE | 6-Amino-2,3-dihydro-phtha...)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125759(5-Amino-2,3-dihydro-phthalazine-1,4-dione | CHEMBL...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125775(2-Amino-8-piperidin-1-yl-1,9-dihydro-purin-6-one |...)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125774(5-Fluoro-1H-indole-2-carboxylic acid hydrazide | C...)
Affinity DataKi:  7.20E+4nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125763(2-BUTYL-5,6-DIHYDRO-1H-IMIDAZO[4,5-D]PYRIDAZINE-4,...)
Affinity DataKi:  8.30E+4nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125770(6-Methyl-2H-pyrazolo[3,4-b]quinolin-3-ylamine | CH...)
Affinity DataKi:  1.56E+5nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125762(5,6-Dihydro-1H-imidazo[4,5-d]pyridazine-4,7-dione ...)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50125764(3-Amino-6-phenyl-2,7-dihydro-pyrazolo[3,4-d]pyrimi...)
Affinity DataKi:  2.49E+5nMAssay Description:Inhibitory activity against eubacterial tRNA guanine transglycosylase (TGT) from Zymomonas mobilisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355756(CHEMBL1909658)
Affinity DataIC50:  13nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355755(CHEMBL1911296)
Affinity DataIC50:  15nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355751(CHEMBL1911286)
Affinity DataIC50:  21nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355758(CHEMBL1911306)
Affinity DataIC50:  139nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355757(CHEMBL1911298)
Affinity DataIC50:  142nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355753(CHEMBL1911289)
Affinity DataIC50:  503nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491557(CHEMBL2046886)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase D516V mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355752(CHEMBL1911287)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50386752(CHEMBL2046887)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase S531L mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355754(CHEMBL1911295)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491558(CHEMBL2046885)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase D516V mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50386752(CHEMBL2046887)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase D516V mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491559(KRM-1648 | Rifalazil)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase S531L mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491558(CHEMBL2046885)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase S531L mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491557(CHEMBL2046886)
Affinity DataIC50:  9.20E+4nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase S531L mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | RIFAMPIN | Rifadin | Rifampic...)
Affinity DataIC50:  1.71E+5nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase S531L mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491559(KRM-1648 | Rifalazil)
Affinity DataIC50:  2.04E+5nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase D516V mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | RIFAMPIN | Rifadin | Rifampic...)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase D516V mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491559(KRM-1648 | Rifalazil)
Affinity DataIC50:  2.99E+5nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase H526Y mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | RIFAMPIN | Rifadin | Rifampic...)
Affinity DataIC50:  1.13E+6nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase H526Y mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50491558(CHEMBL2046885)
Affinity DataIC50:  1.15E+6nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase H526Y mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA-directed RNA polymerase subunit beta(Escherichia coli)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50386752(CHEMBL2046887)
Affinity DataIC50:  1.58E+6nMAssay Description:Inhibition of rifamycin-resistant Escherichia coli RNA polymerase H526Y mutant after 10 mins by rolling circle transcription assay in presence of DNA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355759(CHEMBL1911299)
Affinity DataEC50:  2.10E+3nMAssay Description:Activation of human PXR in DPX2 cells after 24 hrs by microplate reader relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | RIFAMPIN | Rifadin | Rifampic...)
Affinity DataEC50:  5.60E+3nMAssay Description:Activation of human PXR in DPX2 cells after 24 hrs by microplate reader relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50386752(CHEMBL2046887)
Affinity DataEC50:  5.50E+3nMAssay Description:Activation of PXR in human DPX2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | RIFAMPIN | Rifadin | Rifampic...)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of PXR in human DPX2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50355760(CHEMBL1911307)
Affinity DataEC50:  4.10E+3nMAssay Description:Activation of human PXR in DPX2 cells after 24 hrs by microplate reader relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed