Affinity DataKi: 230nMAssay Description:Inhibition of human trypsin and the control activity being 7.3 umol/min/mgMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of EGFR in human A-431 cell membrane vesicles using phospholipase C-gamma-1 as substrate incubated for 10 mins by scintillation counter me...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of ABCG2 (unknown origin)More data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human acrosin and control activity being 11.3 umol/min/mgMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SARS-CoV-2 MProMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SARS-CoV-2 MProMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of SARS-CoV-2 (BetaCoV/Wuhan/WIV04/2019) MPro expressed in Escherichia coli using FRET susbtrate measured after 1 hrMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of EGFR in human A-431 cell membrane vesicles using phospholipase C-gamma-1 as substrate incubated for 10 mins by scintillation counter me...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of human trypsin and the control activity being 7.3 umol/min/mgMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of SARS-CoV-2 MProMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dr. Harisingh Gour University
Curated by ChEMBL
Dr. Harisingh Gour University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant SARS-CoV-2 MPro incubated for 10 mins in presence of fluorogenic substrateMore data for this Ligand-Target Pair