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Found 290 with Last Name = 'giddings' and Initial = 'a'
TargetCoagulation factor X(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307292(2-(2-Carbamimidoyl-benzo[b]thiophen-4-yloxy)-2-phe...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of factor 10a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307291(4-[2-(2-Carbamimidoyl-benzo[b]thiophen-4-yloxy)-2-...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of factor 10a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]neurotensin from rat NTS1 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]neurotensin from rat NTS1 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307314(CHEMBL597557 | [2-Isobutylamino-methyl)-phenyl]-ca...)
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  2nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307290(1-{4-[2-(2-Carbamimidoyl-benzo[b]thiophen-4-yloxy)...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of factor 10a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307267(CHEMBL597759 | [2-(Piperazin-1-ylmethyl)-phenyl]-c...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307308((R)-(4-Methoxy-phenyl)-carbamic acid 2-(2-carbamim...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307313((2-Methylamino-methyl-phenyl)-carbamic acid 2-(2-c...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307277(CHEMBL604954 | [5-(Isopropylamino-methyl)-1,3-dime...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307312((2-Aminomethyl-phenyl)-carbamic acid 2-(2-carbamim...)
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307310(CHEMBL597143 | [4-(2-Dimethylamino-ethoxy)-phenyl]...)
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307279((2-Aminomethyl-phenyl)-carbamic acid 2-(2-carbamim...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307303((2-Fluoro-phenyl)-carbamic acid 2-(2-carbamimidoyl...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307273((5-Methaminomethyl-2-methyl-2H-pyrazol-3-yl)-carba...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307307((4-Methoxy-phenyl)-carbamic acid 2-(2-carbamimidoy...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307276((5-Ethylaminomethyl-1,3-dimethyl-1H-pyrazol-4-yl)-...)
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [125I]neurotensin from rat NTS2 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]NT at rat NTS2 overexpressed in CHOK1 cells after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  7nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 2 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307268((2,4-Difluoro-phenyl)-carbamic acid 2-(2-carbamimi...)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307269((2,6-Difluoro-phenyl)-carbamic acid 2-(2-carbamimi...)
Affinity DataKi:  7nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307306(CHEMBL604289 | o-Tolyl-carbamic acid 2-(2-carbamim...)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307305((4-Fluoro-phenyl)-carbamic acid 2-(2-carbamimidoyl...)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307315((2-Dimethylaminomethyl-phenyl)-carbamic acid 2-(2-...)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307274((3,5-Dimethyl-1H-pyrazol-4-yl)-carbamic acid 2-(2-...)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307280((2-Dimethylaminomethyl-phenyl)-carbamic acid 2-(2-...)
Affinity DataKi:  8.10nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307272((5-Methoxymethyl-2-methyl-2H-pyrazol-3-yl)-carbami...)
Affinity DataKi:  9nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307271((2,5-Dimethyl-2H-pyrazol-3-yl)-carbamic acid 2-(2-...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307311(CHEMBL597144 | [4-(4-Methyl-piperazin-1-ylmethyl)-...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307301(CHEMBL598400 | Phenyl-carbamic acid 2-(2-carbamimi...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307275(CHEMBL601231 | {4-[2-(2-Carbamimidoyl-benzo[b]thio...)
Affinity DataKi:  11nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307270((3,5-Dimethyl-isoxazol-4-yl)-carbamic acid 2-(2-ca...)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307278(CHEMBL602083 | Phenyl-carbamic acid 2-(2-carbamimi...)
Affinity DataKi:  15.5nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]NT at rat NTS2 overexpressed in CHOK1 cells after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  21nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 2 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307304((3-Fluoro-phenyl)-carbamic acid 2-(2-carbamimidoyl...)
Affinity DataKi:  25nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50041429(CHEMBL3356854)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50041428(CHEMBL3356855)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50041427(CHEMBL3356853)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307300(CHEMBL606194 | Ethyl-carbamic acid 2-(2-carbamimid...)
Affinity DataKi:  28nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  28nMAssay Description:Displacement of [125I]neurotensin from rat NTS2 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307297(4-[1-Phenyl-2-(3-phenyl-ureido)-ethoxy]-benzo[b]th...)
Affinity DataKi:  29nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  33nMAssay Description:Displacement of [125I]NT at rat NTS2 overexpressed in CHOK1 cells after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019405(LEVOCABASTINE | R-50547)
Affinity DataKi:  33nMAssay Description:Displacement of [125I]NT at rat NTS2 overexpressed in CHOK1 cells after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307309((S)-(4-Methoxy-phenyl)-carbamic acid 2-(2-carbamim...)
Affinity DataKi:  35nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307296(CHEMBL597370 | [2-(2-Carbamimidoyl-benzo[b]thiophe...)
Affinity DataKi:  50nMAssay Description:Inhibition of human recombinant factor 9a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Trigen

Curated by ChEMBL
LigandPNGBDBM50307289(2-(2-Carbamimidoyl-benzo[b]thiophen-4-yloxy)-N-(4-...)
Affinity DataKi:  52nMAssay Description:Inhibition of factor 10a by amidolytic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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