TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of human KDR/VEGFR2 using poly [Glu:Tyr] as substrate incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liqui...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of human PDGFRa using poly [Glu:Tyr] as substrate incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liquid sc...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of human c-SRC using poly [Glu:Tyr] as substrate incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liquid sci...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of human FGFR1 using KKKSPGEYVNIEFG as substrate incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liquid sci...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK as substrate incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liquid scinti...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Peking Union Medical College And Chinese Academy Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: <10nMAssay Description:Inhibition of human LYN using poly [Glu:Tyr] as substrate incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liquid scint...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of human recombinant DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of rat spinal DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of rat spinal DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of rat spinal DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of rat spinal DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of human recombinant DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of DAAO in porcine kidney homogenate using D-alanine as substrate assessed as pyruvate production incubated for 5 mins by microplate reade...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Chinese Academy Of Medical Sciences&Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human recombinant DAAO using D-alanine as substrate assessed as pyruvate production incubated for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair