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Found 58 with Last Name = 'grant' and Initial = 'mk'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)
Affinity DataKi:  0.129nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)
Affinity DataKi:  2.57nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)
Affinity DataKi:  4.68nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)
Affinity DataKi:  5.25nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)
Affinity DataKi:  5.75nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)
Affinity DataKi:  9.55nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)
Affinity DataKi:  41.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)
Affinity DataKi:  49nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)
Affinity DataKi:  77.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataIC50:  18nMpH: 6.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 6 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003351(3-(4-butoxy-1,2,5-thiadiazol-3-yl)-1-methyl-1,2,5,...)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataIC50:  29nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003366(1-Methyl-5-(4-pentyloxy-[1,2,5]thiadiazol-3-yl)-1,...)
Affinity DataIC50:  33nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072215(1-Methyl-5-[4-(3-phenyl-prop-2-ynyloxy)-[1,2,5]thi...)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003369(1-Methyl-5-(4-propoxy-[1,2,5]thiadiazol-3-yl)-1,2,...)
Affinity DataIC50:  52nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423615(CHEMBL405125)
Affinity DataIC50:  59nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataIC50:  81nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003365(3-(3-(ethoxy)-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetra...)
Affinity DataIC50:  141nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072234(1-Methyl-5-[4-(4-phenyl-butoxy)-[1,2,5]thiadiazol-...)
Affinity DataIC50:  145nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423611(CHEMBL270031)
Affinity DataIC50:  162nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)
Affinity DataIC50:  219nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)
Affinity DataIC50:  275nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423614(CHEMBL403829)
Affinity DataIC50:  309nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)
Affinity DataIC50:  407nMpH: 6.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 6 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423613(CHEMBL271774)
Affinity DataIC50:  617nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423609(CHEMBL406802)
Affinity DataIC50:  646nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423608(CHEMBL272468)
Affinity DataIC50:  871nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423608(CHEMBL272468)
Affinity DataIC50:  871nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataIC50:  955nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423612(CHEMBL406570)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423619(CHEMBL257683)
Affinity DataIC50:  1.07E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423610(CHEMBL255791)
Affinity DataIC50:  1.91E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072215(1-Methyl-5-[4-(3-phenyl-prop-2-ynyloxy)-[1,2,5]thi...)
Affinity DataIC50:  2.14E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423608(CHEMBL272468)
Affinity DataIC50:  2.29E+3nMpH: 6.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 6 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataIC50:  2.40E+3nMpH: 6.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 6 by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423618(CHEMBL401694)
Affinity DataIC50:  3.80E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423609(CHEMBL406802)
Affinity DataIC50:  3.98E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataIC50:  4.90E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423616(CHEMBL272359)
Affinity DataIC50:  7.08E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003366(1-Methyl-5-(4-pentyloxy-[1,2,5]thiadiazol-3-yl)-1,...)
Affinity DataIC50:  8.51E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072234(1-Methyl-5-[4-(4-phenyl-butoxy)-[1,2,5]thiadiazol-...)
Affinity DataIC50:  9.12E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)
Affinity DataIC50:  1.20E+4nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423611(CHEMBL270031)
Affinity DataIC50:  1.48E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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