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Found 1327 with Last Name = 'green' and Initial = 'l'
TargetB2 bradykinin receptor(Cavia porcellus)
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50406750(Firazyr | HOE-140 | Icatibant)
Affinity DataKi:  0.110nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50406751(CHEMBL2369941)
Affinity DataKi:  0.160nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Scios Nova

Curated by ChEMBL
LigandPNGBDBM50406749(CHEMBL2028979)
Affinity DataKi:  0.75nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223637(Alphacemethadone | Alphacetylmethadol)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223633(Levomethadone)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322986(CHEMBL1210141 | N-(1-((2,6-diethoxy-4'-(trifluorom...)
Affinity DataKi:  2.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322979(CHEMBL1210209 | N-(1-((2,6-diethoxy-4'-fluorobiphe...)
Affinity DataKi:  2.5nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223637(Alphacemethadone | Alphacetylmethadol)
Affinity DataKi:  3.40nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322988(CHEMBL1210084 | N-(1-(3,5-diethoxy-4-methylbenzyl)...)
Affinity DataKi:  4nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322987(CHEMBL1210085 | N-(1-(4-chloro-3,5-diethoxybenzyl)...)
Affinity DataKi:  4.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322981(CHEMBL1210207 | N-(1-((2,6-diethoxy-4'-fluorobiphe...)
Affinity DataKi:  4.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322992(CHEMBL1210030 | N-(1-((2-ethoxy-4'-fluorobiphenyl-...)
Affinity DataKi:  4.90nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322980(CHEMBL1210208 | N-(1-((2,6-diethoxybiphenyl-4-yl)m...)
Affinity DataKi:  5.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322984(CHEMBL1210143 | N-(1-(3,5-diethoxy-4-fluorobenzyl)...)
Affinity DataKi:  6.30nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322978(6-amino-N-(1-((2-(benzyloxy)-6-ethoxy-4'-fluorobip...)
Affinity DataKi:  6.70nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322983(CHEMBL1210144 | N-(1-((2,6-diethoxybiphenyl-4-yl)m...)
Affinity DataKi:  6.90nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336997(2-chloro-4-((1R,2S)-1-(5-(4-cyanophenyl)-1,3,4-oxa...)
Affinity DataKi:  7nMAssay Description:Displacement of fluorescent-tagged R1881 from androgen receptor after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19455(4-(3-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-5,7-bis(...)
Affinity DataKi:  7nM ΔG°:  -42.6kJ/mole EC50:  90nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322985(6-amino-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl...)
Affinity DataKi:  7.10nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322982(6-chloro-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-y...)
Affinity DataKi:  7.90nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322971(CHEMBL1210375 | rac-N-(1-((2,6-diethoxy-4'-fluorob...)
Affinity DataKi:  9.30nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataKi:  10nMAssay Description:Displacement of fluorescent-tagged R1881 from androgen receptor after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322991(CHEMBL1210031 | N-(1-((2-ethoxy-4'-(trifluoromethy...)
Affinity DataKi:  11nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322989(CHEMBL1210083 | N-(1-(3,5-diethoxy-4-(1H-imidazol-...)
Affinity DataKi:  11nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227099(2-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-ylami...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223631(Betacetylmethadol)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(CHEMBL241329 | N-(1-(4-chloro-3-ethoxybenzyl)piper...)
Affinity DataKi:  15nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227100(2-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-ylamino)...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322977(CHEMBL1210268 | N-(1-(3,5-diethoxy-4-fluorobenzyl)...)
Affinity DataKi:  18nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322976((R)-N-(1-(4-chloro-3-ethoxybenzyl)azepan-4-yl)-5-m...)
Affinity DataKi:  18nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322993(6-amino-N-(1-(3-ethoxy-4-methylbenzyl)piperidin-4-...)
Affinity DataKi:  19nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227129(CHEMBL241329 | N-(1-(4-chloro-3-ethoxybenzyl)piper...)
Affinity DataKi:  20nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227132(4-tert-butyl-N-(1-((1,4-dimethoxynaphthalen-2-yl)m...)
Affinity DataKi:  20nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322994(CHEMBL1210028 | N-(1-(3-ethoxy-4-methylbenzyl)pipe...)
Affinity DataKi:  21nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322972((R)-N-(1-(3-ethoxy-4-methylbenzyl)azepan-4-yl)-5-m...)
Affinity DataKi:  22nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322974((R)-N-(1-(3,5-diethoxy-4-fluorobenzyl)azepan-4-yl)...)
Affinity DataKi:  22nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227119(CHEMBL236588 | N-(1-(3-isobutoxy-4-methoxybenzyl)p...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322973(CHEMBL1210373 | N-(1-(3,5-diethoxy-4-fluorobenzyl)...)
Affinity DataKi:  25nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19454(4-[2-(4-hydroxyphenyl)-5,7-bis(trifluoromethyl)pyr...)
Affinity DataKi:  26nM ΔG°:  -39.7kJ/mole EC50:  6.00E+3nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataKi:  29nMAssay Description:Displacement of fluorescent-tagged R1881 from androgen receptor after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227117(CHEMBL236611 | N-(1-(3-ethoxy-4-methylbenzyl)piper...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227130(CHEMBL241328 | N-(1-((1,4-dimethoxynaphthalen-2-yl...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19456(4-(3-{4-[2-(dimethylamino)ethoxy]phenyl}-5,7-bis(t...)
Affinity DataKi:  47nM ΔG°:  -38.3kJ/mole EC50:  1.00E+3nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19454(4-[2-(4-hydroxyphenyl)-5,7-bis(trifluoromethyl)pyr...)
Affinity DataKi:  48nM ΔG°:  -38.3kJ/mole EC50:  600nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19453(4-[3-phenyl-5,7-bis(trifluoromethyl)pyrazolo[1,5-a...)
Affinity DataKi:  51nM ΔG°:  -38.1kJ/molepH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227131(CHEMBL241330 | N-(1-(4-chloro-3-ethoxybenzyl)piper...)
Affinity DataKi:  60nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227106(4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)met...)
Affinity DataKi:  66nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University of Illinois At Urbana-Champaign

LigandPNGBDBM19455(4-(3-{4-[2-(piperidin-1-yl)ethoxy]phenyl}-5,7-bis(...)
Affinity DataKi:  71nM ΔG°:  -37.4kJ/mole EC50:  40nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223633(Levomethadone)
Affinity DataKi:  77nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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