Affinity DataKi: 0.110nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:In vitro binding affinity against bradykinin receptor B2 from guinea pig ileum.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of fluorescent-tagged R1881 from androgen receptor after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -42.6kJ/mole EC50: 90nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of fluorescent-tagged R1881 from androgen receptor after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nM ΔG°: -39.7kJ/mole EC50: 6.00E+3nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of fluorescent-tagged R1881 from androgen receptor after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
Affinity DataKi: 47nM ΔG°: -38.3kJ/mole EC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
Affinity DataKi: 48nM ΔG°: -38.3kJ/mole EC50: 600nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
Affinity DataKi: 51nM ΔG°: -38.1kJ/molepH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human SST5RMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nM ΔG°: -37.4kJ/mole EC50: 40nMpH: 7.5 T: 2°CAssay Description:Relative binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer, and purified full-length human ...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair