Affinity DataKi: 0.0000150nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.0000570nMAssay Description:Inhibition of HIV1 protease by fluorescent peptide substrate based assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.00147nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.00800nMAssay Description:Inhibition of HIV1 protease by fluorescent peptide substrate based assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0360nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Binding Affinity of the compound against Growth hormone secretagogue receptor of swine using [35S]-MK-0677 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]estradiol from ERalpha after 4 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity to ERalpha ligand binding domainMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Displacement of [3H]estradiol from ERalpha after 4 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity to ERalpha ligand binding domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]estradiol from ERalpha after 4 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]estradiol from ERbeta after 4 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.780nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine
Curated by ChEMBL
Emory University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.74nMAssay Description:Displacement of [3H]estradiol from ERbeta after 4 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair