Compile Data Set for Download or QSAR
maximum 50k data
Found 19 with Last Name = 'guerra' and Initial = 'l'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254293(CHEMBL4070283)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of BTK in human monocytes assessed as inhibition of FCgammaR activation-induced TNFalpha production by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254289(CHEMBL4091215)
Affinity DataKi:  9.50E+4nMAssay Description:Mixed type inhibition of Electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate after 7 min by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254288(CHEMBL4074057)
Affinity DataKi:  1.06E+5nMAssay Description:Mixed type inhibition of Electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate after 7 min by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029359(4-Amino-2-aminomethyl-3-methyl-butyric acid | CHEM...)
Affinity DataKi:  7.20E+5nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254287(CHEMBL4094588)
Affinity DataKi:  1.57E+6nMAssay Description:Inhibition of BTK in goat anti-human IgM F(ab')2-stimulated human whole blood assessed as suppression of BCR-induced CD69 expression on B cells prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029357(4-Amino-2-aminomethyl-2,3-dimethyl-butyric acid | ...)
Affinity DataKi:  1.65E+6nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029366(4-Amino-2-aminomethyl-butyric acid | CHEMBL139503)
Affinity DataKi:  1.79E+6nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50009385(1,4-butylenediamine | 1,4-tetramethylenediamine | ...)
Affinity DataKi:  3.50E+6nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029364(2,3-dimethyl-1,4-butanediammonium)
Affinity DataKi:  6.10E+6nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029360(2,2-dimethyl-1,4-butanediammonium)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029362(2,2,3-trimethyl-1,4-butanediammonium)
Affinity DataKi: >1.05E+7nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029363(4-Amino-2-aminomethyl-2,3,3-trimethyl-butyric acid...)
Affinity DataKi: >1.10E+7nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029361(2,2,3,3-tetramethyl-1,4-butanediammonium)
Affinity DataKi: >1.10E+7nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029365(4-Amino-2-aminomethyl-3,3-dimethyl-butyric acid | ...)
Affinity DataKi: >1.10E+7nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Rattus norvegicus)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50029358(4-Amino-2-aminomethyl-2-methyl-butyric acid | CHEM...)
Affinity DataKi: >1.10E+7nMAssay Description:Inhibition of liver Ornithine decarboxylase in thioacetamide-treated ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254288(CHEMBL4074057)
Affinity DataIC50:  2.27E+5nMAssay Description:Inhibition of Electric eel AChE using acetylthiocholine as substrate after 7 min by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254289(CHEMBL4091215)
Affinity DataIC50:  4.03E+5nMAssay Description:Mixed type inhibition of Electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate after 7 min by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254293(CHEMBL4070283)
Affinity DataIC50:  9.19E+5nMAssay Description:Inhibition of Electric eel AChE using acetylthiocholine as substrate after 7 min by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50254287(CHEMBL4094588)
Affinity DataIC50:  1.83E+6nMAssay Description:Inhibition of Electric eel AChE using acetylthiocholine as substrate after 7 min by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed