TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 6.60E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes preincubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+4nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes preincubated for 30 minsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.480nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Genentech
Curated by ChEMBL
Genentech
Curated by ChEMBL
Affinity DataIC50: 0.480nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/B(RAT)
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Hoechst Roussel Pgu Cardiovascular Agents
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair