Affinity DataKi: 0.0230nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.47nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.79nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 4.67nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.46nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 34.1nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Antagonist activity at human cloned B1 receptor expressed in african green monkey COS7 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 64.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 119nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Antagonist activity at human cloned B1 receptor expressed in african green monkey COS7 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 237nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Antagonist activity at human cloned B1 receptor expressed in african green monkey COS7 cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 299nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 463nMAssay Description:Antagonist activity at human cloned B1 receptor expressed in african green monkey COS7 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 497nMAssay Description:Antagonist activity at human cloned B1 receptor expressed in african green monkey COS7 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 645nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 654nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 772nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+3nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+3nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.43E+3nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+3nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]desArg from human B1 in human WI 38 cellsMore data for this Ligand-Target Pair