Compile Data Set for Download or QSAR
maximum 50k data
Found 115 with Last Name = 'handlon' and Initial = 'al'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241083(6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1...)
Affinity DataIC50:  0.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199205(6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-6-...)
Affinity DataIC50:  0.740nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199202(6-(4-chlorophenyl)-3-[2-(1-piperidinylmethyl)-6-qu...)
Affinity DataIC50:  0.890nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422940(CHEMBL213008)
Affinity DataIC50:  1nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199219(6-(4-chlorophenyl)-3-[2-(1-pyrrolidinylmethyl)-6-q...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199229(6-(4-chlorophenyl)-3-{2-[(4-phenyl-1-piperidinyl)m...)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422936(CHEMBL212657)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199223(6-(4-chlorophenyl)-3-[2-({4-[2-(1-pyrrolidinyl)eth...)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422927(CHEMBL441368)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422930(CHEMBL214276)
Affinity DataIC50:  2nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199214(6-(4-chlorophenyl)-3-[2-(1H-imidazol-1-ylmethyl)-6...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199206(6-(4-chlorophenyl)-3-[2-(1-pyrrolidinylmethyl)-3,4...)
Affinity DataIC50:  2.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422924(CHEMBL214416)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199240(6-(4-chlorophenyl)-3-(2-{[4-(4-fluorophenyl)-1-pip...)
Affinity DataIC50:  3.10nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199236(6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)m...)
Affinity DataIC50:  3.10nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199204(6-(4-chlorophenyl)-3-{(2R)-2-[(dimethylamino)methy...)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199228(6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-3,...)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422926(CHEMBL215565)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199203(6-(4-chlorophenyl)-3-(2-{[(3R)-3-hydroxy-1-pyrroli...)
Affinity DataIC50:  3.40nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199217(6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)m...)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199212(6-(4-chlorophenyl)-3-[2-(hydroxymethyl)-6-quinolin...)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199215(6-(4-chlorophenyl)-3-{2-[(4-phenyl-1-piperazinyl)m...)
Affinity DataIC50:  3.80nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199216(6-(4-chlorophenyl)-3-[2-(4-morpholinylmethyl)-6-qu...)
Affinity DataIC50:  4.90nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422932(CHEMBL212958)
Affinity DataIC50:  5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422939(CHEMBL439146)
Affinity DataIC50:  5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199234(6-(4-chlorophenyl)-3-(2-{[(3S)-3-hydroxy-1-pyrroli...)
Affinity DataIC50:  5.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199241(6-(4-chlorophenyl)-3-(2-{[4-(1-pyrrolidinyl)-1-pip...)
Affinity DataIC50:  5.60nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199235(6-(4-chlorophenyl)-3-[2-({4-[4-(trifluoromethyl)ph...)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199211(6-(4-chlorophenyl)-3-{2-[(4-ethyl-1-piperazinyl)me...)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422922(CHEMBL384113)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422933(CHEMBL212137)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199209((R)-6-(4-chlorophenyl)-3-(2-(cyclopentylmethyl)-2,...)
Affinity DataIC50:  7nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199239(6-(4-chlorophenyl)-3-{2-[(dimethylamino)methyl]-2,...)
Affinity DataIC50:  7.70nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199207(6-(4-chlorophenyl)-3-[2-(4-morpholinylmethyl)-3,4-...)
Affinity DataIC50:  8.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422938(CHEMBL215862)
Affinity DataIC50:  13nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199208(6-(4-chlorophenyl)-3-[2-({4-[2-(4-morpholinyl)ethy...)
Affinity DataIC50:  19nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422921(CHEMBL214429)
Affinity DataIC50:  20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199233(6-(4-chlorophenyl)-3-(2-{[(2S)-2-(methoxymethyl)py...)
Affinity DataIC50:  24nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199222(6-(4-chlorophenyl)-3-{(2S)-2-[(dimethylamino)methy...)
Affinity DataIC50:  25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422935(CHEMBL215334)
Affinity DataIC50:  25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422929(CHEMBL212883)
Affinity DataIC50:  25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199220(6-[4-(methyloxy)phenyl]-3-[2-(4-morpholinylmethyl)...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199238(3-[2-(4-morpholinylmethyl)-6-quinolinyl]-6-[4-(tri...)
Affinity DataIC50:  36nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199221(6-(4-chlorophenyl)-3-[2-({4-[3-(4-morpholinyl)prop...)
Affinity DataIC50:  37nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199218(6-(4-bromophenyl)-3-[2-(4-morpholinylmethyl)-6-qui...)
Affinity DataIC50:  40nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199231(6-(4-chlorophenyl)-3-(6-quinolinyl)thieno[3,2-d]py...)
Affinity DataIC50:  63nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199224(6-(4-chlorophenyl)-3-(2-{[methyl(phenyl)amino]meth...)
Affinity DataIC50:  87nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422923(CHEMBL387195)
Affinity DataIC50:  100nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422928(CHEMBL214427)
Affinity DataIC50:  126nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199213(6-[4-(1-methylpropyl)phenyl]-3-[2-(4-morpholinylme...)
Affinity DataIC50:  200nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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