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Found 54 with Last Name = 'hatsushiba' and Initial = 'e'
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291167(1-((S)-Oxo-3-(R)-2-amino-1-phenyl-propyl)-pyrrolid...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291175(((R)-1-Benzyl-2-{(S)-2-[(R)-4-guanidino-1-(thiazol...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291175(((R)-1-Benzyl-2-{(S)-2-[(R)-4-guanidino-1-(thiazol...)
Affinity DataIC50:  2nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291173(1-((S)-2-Amino-3-(R)-phenyl-propionyl)-azetidine-2...)
Affinity DataIC50:  3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037610(1-{(S)-2-[(S)-2-(4,5-Dihydro-thiazole-2-carbonyl)-...)
Affinity DataIC50:  3.80nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037612(1-{(S)-2-[(S)-2-(Benzothiazole-2-carbonyl)-pyrroli...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291167(1-((S)-Oxo-3-(R)-2-amino-1-phenyl-propyl)-pyrrolid...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50291163(4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50:  4.40nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50284127(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037605((S)-2-[(S)-2-(Benzothiazole-2-carbonyl)-pyrrolidin...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50291168((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  5nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037611(1-{(S)-2-[(S)-2-(Oxazolo[4,5-b]pyridine-2-carbonyl...)
Affinity DataIC50:  5.5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037606(1-{(S)-2-[(S)-2-(Benzooxazole-2-carbonyl)-pyrrolid...)
Affinity DataIC50:  5.60nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037597(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-4-carbonyl)-pyr...)
Affinity DataIC50:  6.20nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037600(4-Phenyl-1-{(S)-2-[(S)-2-(pyridine-2-carbonyl)-pyr...)
Affinity DataIC50:  6.90nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037609(2-[2-(Thiazole-2-carbonyl)-pyrrolidine-1-carbonyl]...)
Affinity DataIC50:  8.5nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291166((R)-2-((R)-2-Amino-3-phenyl-propionylamino)-N-[(S)...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037602(1-[(S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carbonyl...)
Affinity DataIC50:  8.70nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037604(1-{(S)-2-[(S)-2-(1H-Imidazole-2-carbonyl)-pyrrolid...)
Affinity DataIC50:  9nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291173(1-((S)-2-Amino-3-(R)-phenyl-propionyl)-azetidine-2...)
Affinity DataIC50:  9nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037607(CHEMBL333638 | Oxo-{1-[(S)-1-(4-phenyl-butyryl)-py...)
Affinity DataIC50:  10.3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037603(4-Phenyl-1-{(S)-2-[(S)-2-(pyrimidine-5-carbonyl)-p...)
Affinity DataIC50:  61nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291166((R)-2-((R)-2-Amino-3-phenyl-propionylamino)-N-[(S)...)
Affinity DataIC50:  180nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291171((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  230nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291170((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  230nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291172((S)-1-(3-Phenyl-propionyl)-pyrrolidine-2-carboxyli...)
Affinity DataIC50:  230nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50118724((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataIC50:  260nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataIC50:  600nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291174((S)-1-((R)-2-Amino-3-phenyl-propionyl)-piperidine-...)
Affinity DataIC50:  730nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291172((S)-1-(3-Phenyl-propionyl)-pyrrolidine-2-carboxyli...)
Affinity DataIC50:  820nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037599(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-5-carbonyl)-pyr...)
Affinity DataIC50:  1.09E+3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50118724((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037613(4-Phenyl-1-{(S)-2-[(S)-2-(thiophene-2-carbonyl)-py...)
Affinity DataIC50:  1.26E+3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291171((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037614((S)-2-[(S)-2-(Thiophene-2-carbonyl)-pyrrolidine-1-...)
Affinity DataIC50:  2.02E+3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037608(4-Phenyl-1-{(S)-2-[(S)-2-(pyridine-3-carbonyl)-pyr...)
Affinity DataIC50:  2.29E+3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291170((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291164((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50291163(4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50:  6.02E+3nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50291169((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  7.70E+3nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50291164((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  7.80E+3nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291165((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291165((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037596(1-{(S)-2-[2-(Hydroxy-thiazol-2-yl-methyl)-pyrrolid...)
Affinity DataIC50:  1.61E+4nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50037598(4-Phenyl-1-{(S)-2-[(S)-2-(1H-pyrrole-2-carbonyl)-p...)
Affinity DataIC50:  2.13E+4nMAssay Description:In vitro inhibitory activity against prolyl endopeptidase (PEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50291171((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  2.80E+4nMAssay Description:The compound was tested for the inhibitory activity against prolyl endo peptidase(PEP) enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291174((S)-1-((R)-2-Amino-3-phenyl-propionyl)-piperidine-...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291164((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291163(4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291168((S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carboxylic ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
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