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Found 288 with Last Name = 'hauck' and Initial = 'si'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50292299((5S)-3-(3-fluoro-4-(3-methylisoxazol-5-yl)phenyl)-...)
Affinity DataKi:  420nMAssay Description:Inhibition human liver MAOA activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50292302(CHEMBL390465 | N-(((S)-3-(3-fluoro-4-(3-methylisox...)
Affinity DataKi:  950nMAssay Description:Inhibition human liver MAOA activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50292301((5R)-5-((1H-1,2,3-triazol-1-yl)methyl)-3-(3-fluoro...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition human liver MAOA activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50116067((Linezolid)N-[3-(3-Fluoro-4-morpholin-4-yl-phenyl)...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition human liver MAOA activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50292300((5R)-3-(3-fluoro-4-(3-methylisoxazol-5-yl)phenyl)-...)
Affinity DataKi:  2.26E+4nMAssay Description:Inhibition human liver MAOA activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139408(US8889671, 38)
Affinity DataIC50:  67nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139409(US8889671, 39)
Affinity DataIC50:  97nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160040(US9040528, 173)
Affinity DataIC50:  100nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139407(US8889671, 37)
Affinity DataIC50:  120nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139428(US8889671, 65)
Affinity DataIC50:  120nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139386(US8889671, 15)
Affinity DataIC50:  130nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139388(US8889671, 17 | US8889671, 67)
Affinity DataIC50:  140nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139443(US8889671, 47)
Affinity DataIC50:  150nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139445(US8889671, 55)
Affinity DataIC50:  150nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139434(US8889671, 71)
Affinity DataIC50:  160nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139390(US8889671, 19)
Affinity DataIC50:  160nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139376(US8889671, 5)
Affinity DataIC50:  169nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139416(US8889671, 46)
Affinity DataIC50:  170nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139429(US8889671, 66)
Affinity DataIC50:  170nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139397(US8889671, 26)
Affinity DataIC50:  170nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139441(US8889671, 80)
Affinity DataIC50:  170nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139387(US8889671, 16)
Affinity DataIC50:  190nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160029(US9040528, 165 | US9040528, 165(b))
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159978(US9040528, 120)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160059(US9040528, 104)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160058(US9040528, 103)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159930(US9040528, 82)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159923(US9040528, 75)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159897(BDBM159898 | US9040528, 53)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159849(US9040528, 5)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160047(US9040528, 180)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139419(US8889671, 50)
Affinity DataIC50:  200nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139393(US8889671, 22)
Affinity DataIC50:  210nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139431(US8889671, 68)
Affinity DataIC50:  220nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139404(US8889671, 34)
Affinity DataIC50:  230nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139415(US8889671, 45)
Affinity DataIC50:  260nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139403(US8889671, 33)
Affinity DataIC50:  260nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139396(US8889671, 25)
Affinity DataIC50:  260nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139399(US8889671, 29)
Affinity DataIC50:  270nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139435(US8889671, 72)
Affinity DataIC50:  290nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139412(US8889671, 42)
Affinity DataIC50:  290nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159843(BDBM159925 | US9040528, 2 | US9040528, 2(b))
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159848(US9040528, 4)
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159868(US9040528, 24)
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159891(US9040528, 47)
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159922(US9040528, 74(b))
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159843(BDBM159925 | US9040528, 2 | US9040528, 2(b))
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM159951(US9040528, 95 | US9040528, 95(a))
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160001(US9040528, 142 | US9040528, 142(a))
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM160038(US9040528, 171)
Affinity DataIC50:  300nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/ml of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
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