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Found 539 with Last Name = 'heilmann' and Initial = 'j'
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50392999(CHEMBL2152545)
Affinity DataKi:  12.7nMAssay Description:Time dependent inhibition of equine serum BChE assessed as stability constants of inhibitor-enzyme complex using acetylthiocholine as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataKi:  34nMAssay Description:Time dependent inhibition of Electric eel AChE assessed as stability constants of inhibitor-enzyme complex using acetylthiocholine as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataKi:  41nMAssay Description:Time dependent inhibition of equine serum BChE assessed as stability constants of inhibitor-enzyme complex using acetylthiocholine as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50392998(CHEMBL2152544)
Affinity DataKi:  275nMAssay Description:Time dependent inhibition of equine serum BChE assessed as stability constants of inhibitor-enzyme complex using acetylthiocholine as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50392998(CHEMBL2152544)
Affinity DataKi:  1.12E+3nMAssay Description:Time dependent inhibition of Electric eel AChE assessed as stability constants of inhibitor-enzyme complex using acetylthiocholine as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056333(CHEMBL3322470)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056338(CHEMBL3322475)
Affinity DataKi:  1.27E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Homo sapiens (Human))
Friedrich-Schiller-Universitat Jena

Curated by ChEMBL
LigandPNGBDBM50317180(2-[6-(beta-Carboline-2-ium-2-yl)hexyl]-beta-carbol...)
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]ifenprodil from human NR1-1a/NR2B receptor expressed in mouse L13-E6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50056339(CHEMBL3322476)
Affinity DataKi:  3.10E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in HEK cells at 10 uM after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50317179(2-Methyl-9-[9-(2-methyl-beta-carboline-9-yl)nonyl]...)
Affinity DataIC50:  0.492nMAssay Description:Inhibition of electric eel AChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50317179(2-Methyl-9-[9-(2-methyl-beta-carboline-9-yl)nonyl]...)
Affinity DataIC50:  0.507nMAssay Description:Inhibition of equine serum BChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50317178(2-Methyl-9-[12-(2-methyl-beta-carboline-9-yl)dodec...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of electric eel AChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM9426(CHEMBL258928 | Heterodimeric Tacrine-Based Inhibit...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50396135(CHEMBL2171328)
Affinity DataIC50:  2nMAssay Description:Inhibition of horse AChE by colorimetric Ellman assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50396135(CHEMBL2171328)
Affinity DataIC50:  2.04nMAssay Description:Inhibition of horse AChE by colorimetric Ellman assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50377432(CHEMBL258927)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of electric eel AchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of horse AChE by colorimetric Ellman assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM9426(CHEMBL258928 | Heterodimeric Tacrine-Based Inhibit...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of electric eel AchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50317178(2-Methyl-9-[12-(2-methyl-beta-carboline-9-yl)dodec...)
Affinity DataIC50:  4nMAssay Description:Inhibition of equine serum BChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50377439(CHEMBL257126)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of electric eel AchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5nMAssay Description:Inhibition of equine serum BChE by modified Ellman's methodMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377432(CHEMBL258927)
Affinity DataIC50:  5nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5.13nMAssay Description:Inhibition of horse AChE by colorimetric Ellman assayMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377431(CHEMBL258744)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50261344(CHEMBL466338 | N-(3-{[6-Chloro-2,3-dihydropyrrolo[...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of equine serum BuChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377436(CHEMBL255304)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377439(CHEMBL257126)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377433(CHEMBL258926)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50377436(CHEMBL255304)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of electric eel AchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50377435(CHEMBL256919)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of electric eel AchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50261292(CHEMBL466744 | N-[6-Chloro-2,3-dihydropyrrolo[2,1-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of equine serum BuChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377434(CHEMBL407765)
Affinity DataIC50:  12.3nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50377435(CHEMBL256919)
Affinity DataIC50:  12.7nMAssay Description:Inhibition of equine BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Universit£T W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50160078(CHEMBL3787613)
Affinity DataIC50:  13nMAssay Description:Inhibition of human butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50160078(CHEMBL3787613)
Affinity DataIC50:  14nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50261343(CHEMBL466146 | N-(4-{[6-Chloro-2,3-dihydropyrrolo[...)
Affinity DataIC50:  14nMAssay Description:Inhibition of equine serum BuChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  15.6nMAssay Description:Inhibition of electric eel AChE by colorimetric Ellman assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50317183(2-[11-(beta-Carboline-2-ium-2-yl)undecyl]-beta-car...)
Affinity DataIC50:  18nMAssay Description:Inhibition of equine serum BChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50317192(2-Methyl-9-[5-(2-methyl-beta-carboline-9-yl)pentyl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of equine serum BChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50160250(CHEMBL3785472)
Affinity DataIC50:  21nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50317182(2-[12-(beta-Carboline-2-ium-2-yl)dodecyl]-beta-car...)
Affinity DataIC50:  22nMAssay Description:Inhibition of equine serum BChE by modified Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50160255(CHEMBL3785189)
Affinity DataIC50:  22nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50261345(5-(1,2-Dithiolan-3-yl)-N-[8-(6,7,8,9,10,11-hexahyd...)
Affinity DataIC50:  23nMAssay Description:Inhibition of equine serum BuChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50160077(CHEMBL3785861)
Affinity DataIC50:  23nMAssay Description:Inhibition of equine serum butyrylcholinesterase using butyrylcholine iodide as substrate preincubated for 30 mins followed by substrate addition mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
TBA

Curated by ChEMBL
LigandPNGBDBM50377433(CHEMBL258926)
Affinity DataIC50:  23.6nMAssay Description:Inhibition of electric eel AchE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50497922(CHEMBL3323382)
Affinity DataIC50:  25nMAssay Description:Inhibition of equine serum BChE using ATC iodide substrate by DTNB based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
TBA

Curated by ChEMBL
LigandPNGBDBM50497922(CHEMBL3323382)
Affinity DataIC50:  25nMAssay Description:Inhibition of equine serum BChE using ATC iodide substrate by DTNB based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50261342(CHEMBL469153 | N-(5-{[6-Chloro-2,3-dihydropyrrolo[...)
Affinity DataIC50:  26nMAssay Description:Inhibition of equine serum BuChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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