Affinity DataKi: 38nMAssay Description:Inhibition of human GSK-3beta using biotin-AAEELDSRAGS(PO3H2)PQL as substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Inhibition of GSK-3beta using phospho-glycogen synthase peptide-2 as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 0.813nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 0.820nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 45 mins prior to ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health
Curated by ChEMBL
Centre For Addiction And Mental Health
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 45 mins prior to ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto
Curated by ChEMBL
University Of Toronto
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto
Curated by ChEMBL
University Of Toronto
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto
Curated by ChEMBL
University Of Toronto
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto
Curated by ChEMBL
University Of Toronto
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair