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Found 12 with Last Name = 'hicks' and Initial = 'jw'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataKi:  38nMAssay Description:Inhibition of human GSK-3beta using biotin-AAEELDSRAGS(PO3H2)PQL as substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataKi:  770nMAssay Description:Inhibition of GSK-3beta using phospho-glycogen synthase peptide-2 as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50424227(CHEMBL2314112)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50436356(CHEMBL2396702)
Affinity DataIC50:  0.813nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50436356(CHEMBL2396702)
Affinity DataIC50:  0.820nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM50424227(CHEMBL2314112)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 45 mins prior to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM97458(FAAH Inhibitor, 2g)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Centre For Addiction And Mental Health

Curated by ChEMBL
LigandPNGBDBM97458(FAAH Inhibitor, 2g)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 45 mins prior to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50041003(CHEMBL3354977)
Affinity DataIC50:  47nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50041006(CHEMBL3354980)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50041005(CHEMBL3354979)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50041004(CHEMBL3354978)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant MAO-B by luminescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed