TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Competitive inhibition of recombinant human Cdc25B (351 to 380 residues) assessed as hydrolysis of substrate O-methylfluorescein phosphate by Linewea...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.56nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human influenza A virus A/Aichi/2/1968(H3N2) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.66nMAssay Description:Inhibition of human influenza A virus A/Aichi/2/1968(H3N2) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Miyagi Cancer Center Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Inhibition of CDC25B in presence of 2 mM DTTMore data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of CDC25A in presence of 2 mM DTTMore data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 3.15E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 4.23E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 4.26E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 4.26E+3nMAssay Description:Inhibition of CDC25B in presence of 2 mM DTTMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
Affinity DataIC50: 4.69E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 4.88E+3nMAssay Description:Inhibition of CDC25A in presence of 100 mM DTTMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 5.52E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 5.53E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 5.55E+3nMAssay Description:Inhibition of CDC25A in presence of 100 mM DTTMore data for this Ligand-Target Pair
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 6.22E+3nMAssay Description:Inhibition of CDC25AMore data for this Ligand-Target Pair
Affinity DataIC50: 6.23E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 6.25E+3nMAssay Description:Inhibition of CDC25AMore data for this Ligand-Target Pair
Affinity DataIC50: 6.55E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: 6.77E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair