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Found 216 with Last Name = 'hirai' and Initial = 'g'
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345024((R)-(4-(dodecyloxy)-1-(hydroxymethyl)-3-oxo-1,3-di...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146556(Acetic acid (R)-4-decyloxy-1-hydroxymethyl-3-oxo-1...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146559(But-3-enoic acid (R)-1-acetoxymethyl-1-hydroxymeth...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146558(2,2-Dimethyl-propionic acid (S)-4-dodecyloxy-1-hyd...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146555(Acetic acid (S)-4-decyloxy-1-hydroxymethyl-3-oxo-1...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146561(Acetic acid (R)-4-dodecyloxy-1-hydroxymethyl-3-oxo...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146557(Acetic acid (R)-4-benzyloxy-1-hydroxymethyl-3-oxo-...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146554(CHEMBL102042 | Octanoic acid (S)-2-acetoxy-3-hydro...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50146560(Acetic acid (S)-4-dodecyloxy-1-hydroxymethyl-3-oxo...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345027(((R)-4-(3-((2R,3R,5S,6S)-4-(dodecyloxy)-2,3,5,6-te...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345026((1R,2R,4S,5S)-3-(3-((R)-1-((2-tert-butyl-3,3-dimet...)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50571956(CHEMBL4874608)
Affinity DataKi:  2.60E+3nMAssay Description:Competitive inhibition of recombinant human Cdc25B (351 to 380 residues) assessed as hydrolysis of substrate O-methylfluorescein phosphate by Linewea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345025((R)-(4-(dodecyloxy)-1-(hydroxymethyl)-3-oxo-1,3-di...)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345031(((R)-4-(3-((2R,3S,5R,6S)-4-(dodecyloxy)-2,3,5,6-te...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345030(((R)-4-(3-((2R,3S,5R,6S)-4-(dodecyloxy)-2,3,5,6-te...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345028(((R)-4-(3-((1S,2S,3R,4R,5S,6R)-4-(dodecyloxy)-2,3,...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50345029(((R)-1-(hydroxymethyl)-3-oxo-4-(3-((2R,3S,5R,6S)-2...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Miyagi Cancer Center Research Institute

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  1.56nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Miyagi Cancer Center Research Institute

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human influenza A virus A/Aichi/2/1968(H3N2) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (strain A/Aichi/2/1968 H3N2))
Miyagi Cancer Center Research Institute

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  2.66nMAssay Description:Inhibition of human influenza A virus A/Aichi/2/1968(H3N2) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Miyagi Cancer Center Research Institute

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388826(CHEMBL2062715)
Affinity DataIC50:  740nMAssay Description:Inhibition of CDC25B in presence of 2 mM DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388826(CHEMBL2062715)
Affinity DataIC50:  790nMAssay Description:Inhibition of CDC25A in presence of 2 mM DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388822(CHEMBL2062592)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50012280(CHEMBL3260030)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388821(CHEMBL2062591)
Affinity DataIC50:  1.63E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388809(CHEMBL2062597)
Affinity DataIC50:  2.68E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388824(CHEMBL2062594)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388809(CHEMBL2062597)
Affinity DataIC50:  3.33E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388810(CHEMBL2062598)
Affinity DataIC50:  3.63E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388812(CHEMBL2062707)
Affinity DataIC50:  4.23E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388818(CHEMBL2062712)
Affinity DataIC50:  4.26E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388818(CHEMBL2062712)
Affinity DataIC50:  4.26E+3nMAssay Description:Inhibition of CDC25B in presence of 2 mM DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50012323(CHEMBL3260378)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388823(CHEMBL2062593)
Affinity DataIC50:  4.69E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388807(CHEMBL2062590)
Affinity DataIC50:  4.88E+3nMAssay Description:Inhibition of CDC25A in presence of 100 mM DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388823(CHEMBL2062593)
Affinity DataIC50:  5.13E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388808(CHEMBL2062596)
Affinity DataIC50:  5.13E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388820(CHEMBL2062714)
Affinity DataIC50:  5.19E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388810(CHEMBL2062598)
Affinity DataIC50:  5.52E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388825(CHEMBL2062595)
Affinity DataIC50:  5.53E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388818(CHEMBL2062712)
Affinity DataIC50:  5.55E+3nMAssay Description:Inhibition of CDC25A in presence of 100 mM DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388820(CHEMBL2062714)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388823(CHEMBL2062593)
Affinity DataIC50:  6.22E+3nMAssay Description:Inhibition of CDC25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388814(CHEMBL2062709)
Affinity DataIC50:  6.23E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388810(CHEMBL2062598)
Affinity DataIC50:  6.25E+3nMAssay Description:Inhibition of CDC25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
Shinshu University

Curated by ChEMBL
LigandPNGBDBM50388808(CHEMBL2062596)
Affinity DataIC50:  6.55E+3nMAssay Description:Inhibition of CDC25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388819(CHEMBL2062713)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388813(CHEMBL2062708)
Affinity DataIC50:  6.77E+3nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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