Affinity DataKi: 120nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 1More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 1More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 1More data for this Ligand-Target Pair
Affinity DataKi: 1.47E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase M1a enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 1More data for this Ligand-Target Pair
Affinity DataKi: 2.43E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 1More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 4.83E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 5.78E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 1More data for this Ligand-Target Pair
Affinity DataKi: 9.70E+4nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 1.84E+5nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase Mu 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60E+5nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione-S-transferase A1 enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+5nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKi: 7.10E+5nMAssay Description:Inhibitory activity of the compound was measured on recombinant human Glutathione S-transferase PMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding constant for CDC2L2 kinase domainMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIK3CA kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PRKG1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding constant for ARK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MINK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EGFR(G719S) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.10E+3nMAssay Description:Binding constant for EPHA1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 500nMAssay Description:Binding constant for TYK2(JH2domain-pseudokinase) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 4.30nMAssay Description:Binding constant for HPK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHB3 kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 4.30nMAssay Description:Binding constant for FLT3(D835H) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for EPHA6 kinase domainMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIK3CA(E542K) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ABL1(F317I)-phosphorylated kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Binding constant for CLK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 9.10E+3nMAssay Description:Binding constant for RSK4(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding constant for MET kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2B kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for RSK4(Kin.Dom.2-C-terminal) kinase domainMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIK3CA(H1047Y) kinase domainMore data for this Ligand-Target Pair